SCHEMBL9623732

SCHEMBL9623732

COc1cc2c(cc1OC)C(=S)N(CCCN(C)CCc1ccsc1)C2

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.44
HCN4 Q9Y3Q4 1/20 0.44
CYP3A4 P08684 2/20 0.43
ALOX15 P16050 1/20 0.43
SMPD1 P17405 9/20 0.40
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
BLM P54132 1/20 0.38
PMP22 Q01453 1/20 0.38
ABCB1 P08183 1/20 0.37
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10400846 0.96 MAPT (0.40) MAPTHCN4CYP3A4ALOX15SMPD1
SCHEMBL9624425 0.88 HCN4 (0.51) MAPTHCN4CYP3A4ALOX15SMPD1
Hydrochloric Acid SCHEMBL9625697 0.87 CYP3A4 (0.52) MAPTHCN4CYP3A4ALOX15SMPD1
Hydrochloric Acid SCHEMBL9624321 0.87 CYP3A4 (0.52) MAPTHCN4CYP3A4ALOX15SMPD1
SCHEMBL9625873 0.87 SMPD1 (0.35) MAPTHCN4CYP3A4ALOX15SMPD1
SCHEMBL9624720 0.84 HCN4 (0.46) MAPTHCN4CYP3A4ALOX15SMPD1
SCHEMBL9624538 0.83 BCHE (0.37) SMPD1BCHE
SCHEMBL9624931 0.83 HCN4 (0.46) MAPTHCN4CYP3A4ALOX15SMPD1
SCHEMBL9624761 0.82 HCN4 (0.45) MAPTHCN4CYP3A4ALOX15SMPD1
SCHEMBL9625273 0.82 ALDH1A1 (0.42) MAPTHCN4CYP3A4ALOX15SMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed