SCHEMBL9625873

SCHEMBL9625873

Cc1cc2c(cc1C)C(=S)N(CCCN(C)CCc1ccsc1)C2

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 2/20 0.35
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35
SIGMAR1 Q99720 5/20 0.33
MAPT P10636 1/20 0.32
HCN4 Q9Y3Q4 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
LTA4H P09960 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624476 0.87 MAPT (0.38) SMPD1DRD2DRD3SIGMAR1MAPT
SCHEMBL9623732 0.87 MAPT (0.44) SMPD1MAPTHCN4CYP3A4ALOX15
SCHEMBL9624538 0.86 BCHE (0.37) SMPD1DRD2DRD3SIGMAR1
SCHEMBL9623887 0.83 HDAC6 (0.34) SMPD1DRD2DRD3MAPTHCN4
SCHEMBL10400846 0.82 MAPT (0.40) SMPD1MAPTHCN4CYP3A4ALOX15
SCHEMBL9624963 0.82 HDAC6 (0.34) SMPD1DRD2DRD3SIGMAR1MAPT
SCHEMBL9625068 0.81 HDAC6 (0.35) DRD2DRD3SIGMAR1MAPTHCN4
SCHEMBL9625079 0.81 LMNA (0.39) SMPD1
SCHEMBL9624544 0.81 SIGMAR1 (0.43) DRD2DRD3SIGMAR1CYP3A4LTA4H
SCHEMBL9624961 0.79 LMNA (0.39) DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed