SCHEMBL9623977

SCHEMBL9623977

COc1cc2c(cc1OC)C(=O)N(CCCN(C)Cc1cccnc1)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PDE4D Q08499 4/20 0.42
MAPT P10636 1/20 0.41
HCN4 Q9Y3Q4 1/20 0.41
PDE4A P27815 2/20 0.41
PDE4B Q07343 2/20 0.41
PDE4C Q08493 2/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
MAOB P27338 2/20 0.41
HTR1A P08908 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9625013 0.99 CYP3A4 (0.42) MAOAKDM4EALDH1A1HPGDMAPK1
SCHEMBL9624753 0.91 MAPT (0.45) KDM4EALDH1A1HPGDMAPK1HSD17B10
SCHEMBL9624907 0.91 MAPT (0.49) KDM4EALDH1A1HPGDMAPK1HSD17B10
Hydrochloric Acid SCHEMBL9624866 0.90 CYP3A4 (0.46) KDM4EALDH1A1HPGDMAPK1HSD17B10
SCHEMBL9625065 0.87 CHRNB2 (0.43) KDM4EALDH1A1CHRNB2CHRNA4MAOB
SCHEMBL9625211 0.82 HCN4 (0.57) KDM4EALDH1A1HPGDMAPK1HSD17B10
SCHEMBL9625044 0.82 HCN4 (0.52) KDM4EALDH1A1HPGDMAPK1HSD17B10
Hydrochloric Acid SCHEMBL10646362 0.81 CYP3A4 (0.53) KDM4EALDH1A1HPGDMAPK1HSD17B10
SCHEMBL9624772 0.81 HCN4 (0.48) KDM4EPDE4DMAPTHCN4CYP3A4
Hydrochloric Acid SCHEMBL9624432 0.81 CYP3A4 (0.52) KDM4EALDH1A1HPGDMAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed
EP-0269968-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-06-08 EP disclosed