SCHEMBL9625065

SCHEMBL9625065

Cc1cc2c(cc1C)C(=O)N(CCCN(C)Cc1cccnc1)C2

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.43
CHRNA4 P43681 2/20 0.43
MAOB P27338 4/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ACHE P22303 5/20 0.38
DHPS P49366 1/20 0.38
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624201 0.91 CHRNA7 (0.42) KDM4EALDH1A1DHPS
SCHEMBL10644226 0.91 CHRNA7 (0.40) KDM4EALDH1A1DHPS
SCHEMBL10401085 0.90 KDM4E (0.42) CHRNB2CHRNA4MAOBKDM4EALDH1A1
SCHEMBL9623977 0.87 MAOA (0.43) CHRNB2CHRNA4MAOBKDM4EALDH1A1
Hydrochloric Acid SCHEMBL9625013 0.86 CYP3A4 (0.42) CHRNB2CHRNA4MAOBKDM4EALDH1A1
SCHEMBL9624387 0.81 MAPT (0.39) KDM4EALDH1A1DHPS
SCHEMBL9625087 0.81 MAPT (0.43) KDM4EALDH1A1DHPS
SCHEMBL9624248 0.80 HDAC6 (0.35) MAOBKDM4EALDH1A1
SCHEMBL9624753 0.78 MAPT (0.45) KDM4EALDH1A1LMNA
SCHEMBL9624907 0.78 MAPT (0.49) KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed