SCHEMBL9624316

SCHEMBL9624316

CN(CCCN1CCc2cc3c(cc2C1)OCO3)CCc1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 6/20 0.45
SIGMAR1 Q99720 3/20 0.41
DRD2 P14416 1/20 0.41
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
RECQL P46063 1/20 0.39
LTA4H P09960 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
TSHR P16473 1/20 0.38
PKM P14618 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624254 0.93 GNRHR (0.46) GNRHRCYP2D6CYP2C9CYP2C19TDP1
SCHEMBL9624616 0.88 CYP2D6 (0.44) GNRHRSIGMAR1CYP2D6CYP2C9CYP2C19
SCHEMBL9624992 0.85 ABCB1 (0.52) SIGMAR1TDP1KDM4E
SCHEMBL9625255 0.81 SIGMAR1 (0.45) SIGMAR1DRD2KDM4E
SCHEMBL9624622 0.81 GNRHR (0.46) GNRHRCYP2D6CYP2C9CYP2C19TDP1
SCHEMBL9623814 0.79 SIGMAR1 (0.41) SIGMAR1DRD2KDM4E
SCHEMBL9623969 0.78 GNRHR (0.47) GNRHRCYP2D6CYP2C9CYP2C19TDP1
SCHEMBL9625671 0.78 KDM4E (0.38) GNRHRSIGMAR1KDM4E
SCHEMBL9624797 0.71 PDE10A (0.43) DRD2CYP2D6CYP2C9CYP2C19TDP1
SCHEMBL9624080 0.71 SMN1; SMN2 (0.39) SIGMAR1KDM4EPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed