SCHEMBL9623969

SCHEMBL9623969

CN(CCCN1Cc2cc3c(cc2C1=O)OCO3)CCc1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 3/20 0.47
TERT O14746 1/20 0.43
CYP2D6 P10635 4/20 0.39
CYP2C9 P11712 4/20 0.39
CYP2C19 P33261 4/20 0.39
CYP1A2 P05177 3/20 0.39
CYP3A4 P08684 3/20 0.39
TDP1 Q9NUW8 1/20 0.39
KDM4E B2RXH2 1/20 0.38
TSHR P16473 1/20 0.38
LTA4H P09960 1/20 0.38
RECQL P46063 1/20 0.38
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9624622 0.91 GNRHR (0.46) GNRHRTERTCYP2D6CYP2C9CYP2C19
SCHEMBL9624372 0.86 TERT (0.46) GNRHRTERTCYP2D6CYP2C9CYP2C19
SCHEMBL9624208 0.83 GNRHR (0.33) GNRHRCYP2D6CYP2C9CYP2C19TDP1
SCHEMBL9624254 0.83 GNRHR (0.46) GNRHRTERTCYP2D6CYP2C9CYP2C19
SCHEMBL9623839 0.82 ALDH1A1 (0.41) TDP1KDM4ETSHR
SCHEMBL9624482 0.81 TDP1 (0.34) CYP2D6TDP1
SCHEMBL9625104 0.80 EDNRB (0.35) CYP2D6CYP2C19CYP3A4KDM4ETSHR
SCHEMBL9624619 0.80 SMN1; SMN2 (0.37)
SCHEMBL9624420 0.80 ALDH1A1 (0.36) CYP2D6CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL9624625 0.80 ALDH1A1 (0.41) TDP1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116986-A HETEROAROMATIC AMINE DERIVATIVES DR. KARL THOMAE GMBH (DE) 1992-05-26 US disclosed
US-4912115-A Cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1990-03-27 US disclosed