SCHEMBL9625236

SCHEMBL9625236

C=CC(N)c1ccc(O)cn1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.42
ESR2 Q92731 6/20 0.42
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1853872 0.77 ADRA2A (0.35)
SCHEMBL20741307 0.77 ADRA2A (0.35)
SCHEMBL20741308 0.77 ADRA2A (0.35)
SCHEMBL15332425 0.74 ALDH1A1 (0.35)
SCHEMBL2563540 0.74 ALDH1A1 (0.35)
SCHEMBL15022592 0.74 ESR1 (0.55) ESR1ESR2GRIN2B
SCHEMBL15022591 0.74 ESR1 (0.55) ESR1ESR2GRIN2B
SCHEMBL3722303 0.74 ESR1 (0.55) ESR1ESR2GRIN2B
SCHEMBL2897054 0.70 ESR1 (0.50) ESR1ESR2GRIN2B
SCHEMBL28470383 0.69 MEN1 (0.43) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0241428-B1 USE OF 2-AMINOALKYL-5-PYRIDINOL COMPOUNDS AS NOOTROPICS AND ANTIDEPRESSANTS CIBA-GEIGY AG (CH) 1992-03-18 EP claimed
US-4746670-A Use of 2-aminoalkyl-5-pyridinols as nootropic agents and antidepressants CIBA-GEIGY CORPORATION (US) 1988-05-24 US claimed
EP-0019739-B1 2-AMINOALKYL-5-PYRIDINOLES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM CIBA-GEIGY AG (CH) 1984-07-18 EP claimed
US-4260619-A ANTIISCHEMIC CIBA-GEIGY CORPORATION (US) 1981-04-07 US claimed
EP-0241428-B1 USE OF 2-AMINOALKYL-5-PYRIDINOL COMPOUNDS AS NOOTROPICS AND ANTIDEPRESSANTS CIBA-GEIGY AG (CH) 1992-03-18 EP disclosed
US-4746670-A Use of 2-aminoalkyl-5-pyridinols as nootropic agents and antidepressants CIBA-GEIGY CORPORATION (US) 1988-05-24 US disclosed
US-4746670-A Use of 2-aminoalkyl-5-pyridinols as nootropic agents and antidepressants CIBA-GEIGY CORPORATION (US) 1988-05-24 US disclosed
EP-0241428-A2 Use of 2-aminoalkyl-5-pyridinol compounds as nootropics and antidepressants CIBA-GEIGY AG (CH) 1987-10-14 EP disclosed
US-4260619-A ANTIISCHEMIC CIBA-GEIGY CORPORATION (US) 1981-04-07 US disclosed
US-4260619-A ANTIISCHEMIC CIBA-GEIGY CORPORATION (US) 1981-04-07 US disclosed
US-4260619-A ANTIISCHEMIC CIBA-GEIGY CORPORATION (US) 1981-04-07 US disclosed