SCHEMBL9628115

SCHEMBL9628115

COc1ccc2c(c1)CC(CC(=O)O)O2

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.57
GABRA1 P14867 1/20 0.52
GABRB2 P47870 1/20 0.52
MIF P14174 1/20 0.49
MTNR1A P48039 4/20 0.48
ATM Q13315 1/20 0.47
GLS O94925 2/20 0.46
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
TP53 P04637 2/20 0.45
LMNA P02545 1/20 0.45
ABCB1 P08183 1/20 0.44
AR P10275 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
PPARD Q03181 1/20 0.43
FFAR1 O14842 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10257134 0.88 HRH3 (0.60) HRH3GABRA1GABRB2MIFMTNR1A
SCHEMBL17761389 0.88 HRH3 (0.56) HRH3GABRA1GABRB2MTNR1AGLS
SCHEMBL13802286 0.86 FFAR1 (0.56) HRH3GABRA1GABRB2MTNR1AGLS
Hydrochloric Acid SCHEMBL9118102 0.83 HRH3 (0.49) HRH3GABRA1GABRB2MTNR1AGLS
SCHEMBL10256487 0.82 HRH3 (0.59) HRH3GABRA1GABRB2MTNR1AGLS
SCHEMBL7297149 0.81 GABRA1 (0.47) HRH3GABRA1GABRB2MIFMTNR1A
SCHEMBL30637096 0.80 ATM (0.60) MIFMTNR1AATMLMNAABCB1
SCHEMBL9117533 0.80 HRH3 (0.63) HRH3GABRA1GABRB2MTNR1AGLS
SCHEMBL14457195 0.79 FFAR1 (0.42) HRH3ITGB3ITGA2BTP53PPARD
SCHEMBL7289417 0.78 GLS (0.57) HRH3GABRA1GABRB2MTNR1AGLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed