SCHEMBL9628700

SCHEMBL9628700

CCCNC(=O)Oc1ccc2c(c1)C(CN(C)CCC)CO2

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ACHE P22303 16/20 0.49
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10460567 0.83 ACHE (0.48) ACHE
SCHEMBL9628413 0.82 BCHE (0.46) ACHE
Oxalic Acid SCHEMBL9628716 0.81 ACHE (0.46) ACHE
SCHEMBL9628688 0.80 HTR2B (0.43) MTNR1A
SCHEMBL9628703 0.78 ACHE (0.45) ACHE
SCHEMBL9628089 0.78 ACHE (0.41) ACHEMTNR1AMTNR1B
SCHEMBL9628742 0.75 TP53 (0.41) ACHE
Oxalic Acid SCHEMBL9628990 0.75 ACHE (0.39) ACHEMTNR1AMTNR1B
SCHEMBL9627834 0.75 DRD3 (0.45)
SCHEMBL9627777 0.74 PPARG (0.37) ACHEMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP disclosed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP disclosed