SCHEMBL9628089

SCHEMBL9628089

CCCN(CCC)CC1COc2ccc(OC(=O)NC(C)C)cc21

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.41
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
MMP2 P08253 1/20 0.35
CYP3A4 P08684 1/20 0.34
KMT2A Q03164 1/20 0.34
PSMB5 P28074 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL9628990 0.97 ACHE (0.39) ACHEMTNR1AMTNR1BMMP2CYP3A4
SCHEMBL9627808 0.85 BCHE (0.47) ACHE
SCHEMBL9628742 0.83 TP53 (0.41) ACHECYP3A4
SCHEMBL10460567 0.83 ACHE (0.48) ACHE
SCHEMBL9627777 0.82 PPARG (0.37) ACHEMTNR1AMTNR1BKMT2A
Oxalic Acid SCHEMBL9628716 0.81 ACHE (0.46) ACHE
SCHEMBL9627910 0.79 HTR1A (0.44) CYP3A4KMT2A
SCHEMBL9627868 0.78 KMT2A (0.41) KMT2A
SCHEMBL9628700 0.78 ACHE (0.49) ACHEMTNR1AMTNR1B
SCHEMBL10460150 0.78 ACHE (0.39) ACHEMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281261-B1 3-AMINOMETHYL DERIVATIVES OF INDANE, INDOLINE AND DIHYDROBENZOFURANE AND DIHYDROBENZOTHIOPHENE H. LUNDBECK A/S (DK) 1992-05-06 EP claimed
EP-0281261-A2 3-Aminomethyl derivatives of indane, indoline and dihydrobenzofurane and dihydrobenzothiophene H. LUNDBECK A/S (DK) 1988-09-07 EP claimed
US-4946863-A CNS-affecting 6-oxy-3-aminomethyl indanes, compositions thereof, and method of treating therewith H. LUNDBECK A/S (DK) 1990-08-07 US disclosed
US-4847254-A CNS affecting 5-oxy-3-aminomethyl-dihydro-benzofurans and benzothiophenes H. LUNDBECK A/S (DK) 1989-07-11 US disclosed