SCHEMBL9629478

SCHEMBL9629478

Cc1ccc(Cn2c(NC3CCCNCC3)nc3ccccc32)o1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.58
NR4A2 P43354 1/20 0.58
TSHR P16473 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SOS1 Q07889 1/20 0.43
SSTR5 P35346 5/20 0.43
HTT P42858 2/20 0.42
GSK3B P49841 1/20 0.41
TRPC5 Q9UL62 1/20 0.39
LMNA P02545 2/20 0.39
GAA P10253 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CHEK2 O96017 1/20 0.39
MEN1 O00255 1/20 0.39
MLNR O43193 1/20 0.39
CACNA1F O60840 1/20 0.39
EED O75530 1/20 0.39
USP2 O75604 1/20 0.39
ABCB11 O95342 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9697200 0.96 KCNH2 (0.62) KCNH2NR4A2TSHRNPC1RAB9A
Fumaric Acid SCHEMBL9631572 0.92 KCNH2 (0.51) KCNH2NR4A2TSHRNPC1RAB9A
Hydrochloric Acid SCHEMBL9631713 0.89 KCNH2 (0.54) KCNH2NR4A2TSHRNPC1RAB9A
SCHEMBL9630126 0.88 KCNH2 (0.44) KCNH2NR4A2TSHRNPC1RAB9A
SCHEMBL14198334 0.84 TSHR (0.52) KCNH2NR4A2TSHRNPC1RAB9A
SCHEMBL6996422 0.84 KCNH2 (0.62) KCNH2NR4A2SOS1SSTR5HTT
SCHEMBL10397086 0.83 KCNH2 (0.47) KCNH2NR4A2TSHRNPC1RAB9A
Water SCHEMBL9876754 0.82 KCNH2 (0.46) KCNH2NR4A2TSHRNPC1RAB9A
Water SCHEMBL9876758 0.82 KCNH2 (0.46) KCNH2NR4A2TSHRNPC1RAB9A
SCHEMBL9303969 0.82 KCNH2 (0.60) KCNH2NR4A2SOS1SSTR5HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5151424-A Antiallergens or antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-29 US disclosed
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed
US-5071846-A Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1991-12-10 US disclosed
US-4988689-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-01-29 US disclosed
EP-0297661-A1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1989-01-04 EP disclosed