SCHEMBL9630764

SCHEMBL9630764

CC1CC(C)(C)CC(c2ccc(Oc3ccccc3C#N)cc2)(c2ccc(Oc3ccccc3C#N)cc2)C1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
GAA P10253 1/20 0.50
ESR1 P03372 1/20 0.49
ESR2 Q92731 1/20 0.49
EZH2 Q15910 11/20 0.46
KCNH2 Q12809 1/20 0.39
MAPK14 Q16539 2/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
AR P10275 1/20 0.36
LPAR1 Q92633 1/20 0.35
LPAR5 Q9H1C0 1/20 0.35
CYP3A4 P08684 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10112879 0.82 ESR1 (0.45) POLBGAAESR1ESR2EZH2
SCHEMBL8993553 0.81 ESR1 (0.52) GAAESR1ESR2CYP3A4
SCHEMBL9846995 0.80 ESR1 (0.50) ESR1ESR2KCNH2CYP3A4SLC6A4
SCHEMBL9846972 0.78 ESR1 (0.51) POLBGAAESR1ESR2KCNH2
SCHEMBL17042465 0.77 ESR1 (0.59) ESR1ESR2CYP3A4
SCHEMBL9846977 0.74 POLB (0.56) POLBGAAESR1ESR2EZH2
SCHEMBL10000525 0.73 ESR1 (0.66) GAAESR1ESR2
SCHEMBL827205 0.73 ESR1 (0.69) ESR1ESR2CYP3A4
SCHEMBL9472412 0.71 ESR1 (0.67) ESR1ESR2CYP3A4
SCHEMBL3421693 0.71 POLB (0.79) POLBGAAEZH2KCNH2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5105004-A For the preparation of heat stable plastics BAYER AKTIENGESELLSCHAFT (DE) 1992-04-14 US disclosed
EP-0413233-A2 Copolyamides with higher glas transition temperature BAYER AG (DE) 1991-02-20 EP disclosed
EP-0379006-A2 Aminoarylethers BAYER AG (DE) 1990-07-25 EP disclosed
EP-0363760-A1 Aromatic ethers BAYER AG (DE) 1990-04-18 EP disclosed