SCHEMBL10000525

SCHEMBL10000525

COc1ccc(C2(c3ccc(OC)cc3)CC(C)CC(C)(C)C2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.66
ESR2 Q92731 1/20 0.66
MAOB P27338 2/20 0.45
MAOA P21397 1/20 0.45
CHRNA1 P02708 1/20 0.39
CHRNG P07510 1/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
CHRND Q07001 1/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25986540 0.95 ESR1 (0.60) ESR1ESR2MAOBMAOACHRNA1
SCHEMBL12177591 0.93 ESR2 (0.80) ESR1ESR2MAOBMAOACHRNA1
SCHEMBL13382522 0.90 ESR1 (0.55) ESR1ESR2MAOBMAOAKMT2A
SCHEMBL10175309 0.90 ESR1 (0.55) ESR1ESR2MAOBMAOACHRNA1
SCHEMBL22651381 0.88 ESR1 (0.56) ESR1ESR2MAOBMAOACHRNA1
SCHEMBL12021689 0.88 ESR1 (0.56) ESR1ESR2MAOBMAOACHRNA1
SCHEMBL18230813 0.85 PKM (0.51) ESR1ESR2MAOBMAOAKMT2A
SCHEMBL17081749 0.85 ESR1 (0.50) ESR1ESR2MAOBMAOACHRNA1
SCHEMBL23969898 0.84 ESR1 (0.52) ESR1ESR2KMT2AMEN1ALDH1A1
SCHEMBL14516673 0.84 ESR1 (0.49) ESR1ESR2MAOBMAOAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230235115-A1 ESTER COMPOUND AND RESIN COMPOSITION AJINOMOTO CO., INC. (JP) 2023-07-27 US disclosed
US-20230235115-A1 ESTER COMPOUND AND RESIN COMPOSITION AJINOMOTO CO., INC. (JP) 2023-07-27 US disclosed
US-20200148848-A1 POLYCARBONATE COMPOSITE HAVING AN INCREASED PENCIL HARDNESS COVESTRO DEUTSCHLAND AG (DE) 2020-05-14 US disclosed
US-10031430-B2 Electrophotographic photosensitive member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2018-07-24 US disclosed
US-20180173121-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2018-06-21 US disclosed
US-9971257-B2 Electrophotographic photosensitive member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2018-05-15 US disclosed
US-20170343909-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2017-11-30 US disclosed
US-9783673-B2 High-temperature (co)polycarbonates with improved rheological properties COVESTRO DEUTSCHLAND AG (DE) 2017-10-10 US disclosed
US-9783673-B2 High-temperature (co)polycarbonates with improved rheological properties COVESTRO DEUTSCHLAND AG (DE) 2017-10-10 US disclosed
US-20170242350-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2017-08-24 US disclosed
US-20160040009-A1 HIGH-TEMPERATURE (CO)POLYCARBONATES WITH IMPROVED RHEOLOGICAL PROPERTIES COVESTRO DEUTSCHLAND AG (DE) 2016-02-11 US disclosed
US-9139730-B2 (Co)polycarbonates with improved optical properties BAYER MATERIALSCIENCE AG (DE) 2015-09-22 US disclosed
US-9139730-B2 (Co)polycarbonates with improved optical properties BAYER MATERIALSCIENCE AG (DE) 2015-09-22 US disclosed
EP-2313456-B1 MODIFIED POLYCARBONATES HAVING IMPROVED SURFACE PROPERTIES BAYER MATERIALSCIENCE AG (DE) 2013-01-30 EP disclosed
US-20120052412-A1 POLYARYLENE BLOCK COPOLYMER HAVING SULFONIC ACID GROUP AND USE THEREOF HONDA MOTOR CO., LTD. (JP) 2012-03-01 US disclosed
US-20120052412-A1 POLYARYLENE BLOCK COPOLYMER HAVING SULFONIC ACID GROUP AND USE THEREOF HONDA MOTOR CO., LTD. (JP) 2012-03-01 US disclosed
US-20120022204-A1 (CO)POLYCARBONATES WITH IMPROVED OPTICAL PROPERTIES BAYER MATERIALSCIENCE AG (DE) 2012-01-26 US disclosed
US-20120022204-A1 (CO)POLYCARBONATES WITH IMPROVED OPTICAL PROPERTIES BAYER MATERIALSCIENCE AG (DE) 2012-01-26 US disclosed
US-20090245867-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, ELECTROPHOTOGRAPHIC PHOTORECEPTOR CARTRIDGE, AND IMAGE FORMING APPARATUS MITSUBISHI CHEMICAL CORPORATION (JP) 2009-10-01 US disclosed
US-20090245867-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, ELECTROPHOTOGRAPHIC PHOTORECEPTOR CARTRIDGE, AND IMAGE FORMING APPARATUS MITSUBISHI CHEMICAL CORPORATION (JP) 2009-10-01 US disclosed