SCHEMBL9632119

SCHEMBL9632119

COCc1ccsc1C=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 2/20 0.33
PRKCE Q02156 3/20 0.32
MYLK Q15746 2/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PRKCG P05129 1/20 0.32
MAPT P10636 1/20 0.32
PRKCA P17252 1/20 0.32
APEX1 P27695 1/20 0.32
RECQL P46063 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HSD17B3 P37058 1/20 0.32
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
AR P10275 1/20 0.32
CYP2A6 P11509 1/20 0.32
DPP4 P27487 1/20 0.31
TRIM24 O15164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12063377 0.85 CYP2A6 (0.30) CYP2A6
SCHEMBL2065835 0.79
SCHEMBL28271068 0.77 CHRM2 (0.38) SLC6A1L3MBTL1
SCHEMBL14560391 0.75 NQO1 (0.33) MEN1ALDH1A1MAPTKMT2APKM
SCHEMBL1124902 0.75 ALDH1A1 (0.39) MEN1ALDH1A1MAPTKMT2ANPC1
SCHEMBL6816923 0.74 PRKCI (0.33) MEN1KMT2ANPC1PKMRAB9A
SCHEMBL1491977 0.74
SCHEMBL255742 0.74
SCHEMBL3716800 0.74
SCHEMBL9632650 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109206417-B Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2023-01-03 CN disclosed
CN-115124520-A Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2022-09-30 CN disclosed
CN-109206417-A Opioid receptor agonists and uses thereof 四川海思科制药有限公司 2019-01-15 CN disclosed
US-5120861-A DIAZIRINE DERIVATIVES OF AROMATIC HETEROCYCLIC COMPOUNDS SHELL RESEARCH LIMITED (GB) 1992-06-09 US disclosed
EP-0432817-A1 Diazirine derivatives of aromatic heterocyclic compounds SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-06-19 EP disclosed