SCHEMBL9633240

SCHEMBL9633240

CCCCC#C/C=C/CN(C)Cc1cccc2ccccc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.65
LMNA P02545 4/20 0.65
SLC6A2 P23975 3/20 0.65
SIGMAR1 Q99720 3/20 0.65
ADRA2A P08913 2/20 0.65
SQLE Q14534 1/20 0.65
CYP1A2 P05177 2/20 0.58
CYP2C19 P33261 2/20 0.58
NR1I2 O75469 2/20 0.58
HTR2A P28223 2/20 0.58
SLC6A4 P31645 2/20 0.58
KCNH2 Q12809 2/20 0.58
HTT P42858 2/20 0.58
KMT2A Q03164 2/20 0.58
DRD2 P14416 1/20 0.58
ADRA2C P18825 1/20 0.58
CNR1 P21554 1/20 0.58
ADRA1A P35348 1/20 0.58
OPRK1 P41145 1/20 0.58
SLC6A3 Q01959 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9633247 1.00 CYP2D6 (0.65) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL14340050 0.85 CYP2D6 (0.58) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL13407742 0.82 CYP2D6 (0.74) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL10610928 0.82 CYP2D6 (0.60) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL9633950 0.82 CYP2D6 (0.60) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL10610435 0.81 ALDH1A1 (0.43) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL9633517 0.81 ALDH1A1 (0.43) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL9633516 0.81 ALDH1A1 (0.43) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL11006133 0.79 LMNA (0.70) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL9633225 0.79 LMNA (0.70) CYP2D6LMNASLC6A2SIGMAR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4755534-A Propenylamines, pharmaceutical compositions containing them and their use as pharmaceuticals SANDOZ LTD. (CH) 1988-07-05 US claimed
EP-0024587-B1 PROPENYLAMINES, PROCESSES FOR THEIR PRODUCTION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS PHARMACEUTICALS SANDOZ AG (CH) 1984-11-14 EP claimed
US-5132459-A Fungicides SANDOZ LTD. (CH) 1992-07-21 US disclosed
US-4755534-A Propenylamines, pharmaceutical compositions containing them and their use as pharmaceuticals SANDOZ LTD. (CH) 1988-07-05 US disclosed
EP-0024587-B1 PROPENYLAMINES, PROCESSES FOR THEIR PRODUCTION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS PHARMACEUTICALS SANDOZ AG (CH) 1984-11-14 EP disclosed
EP-0024587-A1 Propenylamines, processes for their production, pharmaceutical compositions containing them and their use as pharmaceuticals SANDOZ AG (CH) 1981-03-11 EP disclosed