SCHEMBL9633943

SCHEMBL9633943

CC(=O)c1c(C)c(F)c(F)c(F)c1C

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.39
CYP1A2 P05177 1/20 0.39
TAS1R3 Q7RTX0 11/20 0.38
TAS1R1 Q7RTX1 10/20 0.38
TAS1R2 Q8TE23 10/20 0.38
HSD17B10 Q99714 1/20 0.35
BRD4 O60885 1/20 0.33
BRPF1 P55201 1/20 0.33
CREBBP Q92793 1/20 0.33
THRB P10828 1/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
PKM P14618 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9608357 0.92 TAS1R3 (0.41) CYP3A4CYP1A2TAS1R3TAS1R1TAS1R2
SCHEMBL18674532 0.86 TAS1R3 (0.41) CYP3A4CYP1A2TAS1R3TAS1R1TAS1R2
SCHEMBL13125484 0.84 TAS1R3 (0.44) CYP3A4CYP1A2TAS1R3TAS1R1TAS1R2
SCHEMBL6727338 0.83 TAS1R3 (0.47) CYP3A4CYP1A2TAS1R3TAS1R1TAS1R2
SCHEMBL823811 0.79 CES2 (0.42) CYP3A4CYP1A2THRBMEN1HPGD
SCHEMBL124392 0.79 CES2 (0.42) CYP3A4CYP1A2THRBMEN1HPGD
SCHEMBL19360080 0.79 CES2 (0.42) CYP3A4CYP1A2THRBMEN1HPGD
SCHEMBL19149846 0.78 CYP3A4 (0.48) CYP3A4CYP1A2HSD17B10BRD4BRPF1
SCHEMBL2011531 0.78 MEN1 (0.46) CYP1A2TAS1R3TAS1R1TAS1R2MEN1
SCHEMBL29042640 0.76 CYP3A4 (0.39) CYP3A4CYP1A2HSD17B10THRBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298020-B1 USE OF AN EPOXIDATION REAGENT, AND PROCESS FOR THE PREPARATION OF 5-ALPHA (10-ALPHA) EPOXY-DELTA 9(11) STEROIDS SCHERING AKTIENGESELLSCHAFT (DE) 1992-06-24 EP disclosed