SCHEMBL9635012

SCHEMBL9635012

COC(=O)c1ccc(CC2=CCc3ccc(NC(=O)C(F)(F)F)cc32)c(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
NQO2 P16083 1/20 0.46
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
NPY5R Q15761 1/20 0.39
MAPT P10636 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NR1H4 Q96RI1 2/20 0.37
CYSLTR2 Q9NS75 2/20 0.37
CYSLTR1 Q9Y271 2/20 0.37
EPHX2 P34913 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9634205 0.83 CYSLTR2 (0.53) CYP1A2CYP2C19MEN1KMT2ACYSLTR2
SCHEMBL9647175 0.81 MAPT (0.44) NQO2MTNR1AMTNR1BMAPTMEN1
Hydrochloric Acid SCHEMBL9635452 0.80 MAPT (0.43) NQO2MTNR1AMTNR1BMAPTMEN1
SCHEMBL9635034 0.75 CYSLTR2 (0.62) MEN1KMT2ACYSLTR2CYSLTR1
SCHEMBL9634711 0.73 NQO2 (0.41) CYP1A2CYP2C9CYP2C19NQO2MTNR1A
SCHEMBL9634219 0.73 MEN1 (0.35) NQO2MTNR1AMTNR1BMAPTMEN1
SCHEMBL9635481 0.70 CYP1A2 (0.46) CYP1A2CYP2C9CYP2C19MAPTMEN1
SCHEMBL9634778 0.68 NQO2 (0.40) CYP1A2CYP2C9CYP2C19NQO2MTNR1A
SCHEMBL1542356 0.68 MEN1 (0.61) CYP1A2CYP2C9CYP2C19MAPTMEN1
SCHEMBL6422179 0.66 CYP1A2 (0.73) CYP1A2CYP2C9CYP2C19NPY5RMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337765-B1 ACYLSULFONAMIDE DERIVATIVES OF ALPHA-CARBOCYCLYLTOLUIC ACIDS USED AS LEUKOTRIENE ANTAGONISTS ICI AMERICAS INC. (US) 1992-10-14 EP disclosed
US-5095038-A Antiinflammatory, antiallergens ICI AMERICAS INC. (US) 1992-03-10 US disclosed
EP-0337765-A2 Acylsulfonamide derivatives of alpha-carbocyclyltoluic acids used as leukotriene antagonists ICI AMERICAS INC. (US) 1989-10-18 EP disclosed