SCHEMBL9636604

SCHEMBL9636604

CCN1CCSc2ccccc2C1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RYR2 Q92736 8/20 0.54
KDM1A O60341 2/20 0.40
NOTUM Q6P988 1/20 0.38
KCNH2 Q12809 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
CHRNA7 P36544 1/20 0.37
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15936060 0.83 ALDH1A1 (0.58) RYR2KDM1AALDH1A1CYP1A2CYP2D6
SCHEMBL6867057 0.80 RYR2 (0.51) RYR2KCNH2SIGMAR1
SCHEMBL13622141 0.80 RYR2 (0.55) RYR2NOTUMKCNH2ALDH1A1
SCHEMBL14862467 0.79 RYR2 (0.50) RYR2KDM1ANOTUMKCNH2ALDH1A1
SCHEMBL13622143 0.78 RYR2 (0.60) RYR2NOTUMKCNH2ALDH1A1
SCHEMBL2062177 0.78 RYR2 (0.41) RYR2
SCHEMBL8248175 0.77 RYR2 (0.57) RYR2KDM1ANOTUMKCNH2CYP2D6
SCHEMBL15936312 0.76 RYR2 (0.51) RYR2NOTUMKCNH2SIGMAR1
SCHEMBL15935957 0.76 DRD4 (0.51) RYR2KCNH2ALDH1A1SIGMAR1
SCHEMBL7558332 0.76 RYR2 (0.53) RYR2NOTUMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2764867-A1 Agents for preventing and treating disorders Involving modulation of the RYR receptors The Trustees of Columbia University in the City of New York (US) 2014-08-13 EP claimed
EP-0368063-B1 PROCESS FOR THE CHLORINATION IN THE NUCLEUS OF AROMATIC HYDROCARBONS BAYER AG (DE) 1992-06-10 EP disclosed
US-4990707-A Process for the ring chlorination of aromatic hydrocarbons BAYER AKTIENGESELLSCHAFT (DE) 1991-02-05 US disclosed
EP-0368063-A1 Process for the chlorination in the nucleus of aromatic hydrocarbons BAYER AG (DE) 1990-05-16 EP disclosed