SCHEMBL9639488

SCHEMBL9639488

COC1=CC(=O)OC1C(OC(=O)[C@@H]1CCCN1)c1ccccc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 1/20 0.35
ELANE P08246 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
IDO1 P14902 1/20 0.33
HTR2C P28335 1/20 0.33
HPGD P15428 1/20 0.33
WNT3 P56703 2/20 0.33
SFRP1 Q8N474 2/20 0.33
SLC6A9 P48067 2/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
TACR1 P25103 1/20 0.33
HCRTR2 O43614 1/20 0.32
PDE4D Q08499 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL10394849 0.99 CYP1A2 (0.35) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
SCHEMBL9639322 0.89 CYP3A4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
Bromide SCHEMBL10393939 0.88 CYP3A4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
SCHEMBL9640466 0.88 CYP3A4 (0.37) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
SCHEMBL9640340 0.87 CYP3A4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
SCHEMBL9639485 0.87 CYP3A4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
Hydrochloric Acid SCHEMBL10394208 0.86 CYP3A4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
Bromide SCHEMBL10393772 0.86 CYP3A4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
Bromide SCHEMBL10393773 0.86 CYP3A4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19ELANE
SCHEMBL9640335 0.85 CYP3A4 (0.45) CYP1A2CYP3A4CYP2D6CYP2C19ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0349609-B1 AMINOACID ESTERS, PROCESS FOR THEIR MANUFACTURE AND THEIR USE Dr. Willmar Schwabe GmbH & Co. (DE) 1992-08-05 EP disclosed
WO-1989004310-A1 AMINOACID ESTERS, PROCESS FOR THEIR MANUFACTURE AND THEIR USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1989-05-18 WO disclosed