SCHEMBL9639628

SCHEMBL9639628

CCNc1cccnc1N1CCN(CCOC(C)=O)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.49
CHIA Q9BZP6 1/20 0.46
SLC18A3 Q16572 1/20 0.43
DRD2 P14416 2/20 0.41
HRH3 Q9Y5N1 6/20 0.41
HTR1A P08908 2/20 0.40
HTR2A P28223 1/20 0.40
DRD4 P21917 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
HTR7 P34969 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9755197 0.99 PARP1 (0.48) PARP1CHIASLC18A3DRD2HRH3
SCHEMBL9640183 0.85 SIRT6 (0.47) PARP1CHIADRD2HTR1AHTR2A
Hydrochloric Acid SCHEMBL9639460 0.84 SIRT6 (0.46) PARP1CHIADRD2HTR1AHTR2A
SCHEMBL9639544 0.83 PARP1 (0.50) PARP1CHIADRD2HTR1ADRD4
SCHEMBL9639591 0.82 PARP1 (0.50) PARP1CHIADRD4
Hydrochloric Acid SCHEMBL9640177 0.81 PARP1 (0.49) PARP1CHIADRD4
SCHEMBL9755222 0.81 PARP1 (0.52) PARP1CHIAHTR1A
SCHEMBL9640631 0.80 PARP1 (0.53) PARP1CHIA
SCHEMBL9639730 0.80 PARP1 (0.48) PARP1CHIADRD2HTR1AHTR2A
Fumaric Acid SCHEMBL9755189 0.79 PARP1 (0.48) PARP1CHIADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991006542-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1991-05-16 WO claimed
EP-0496746-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1992-08-05 EP disclosed
WO-1991006542-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1991-05-16 WO disclosed