SCHEMBL964036

SCHEMBL964036

CC(C)NC(=O)c1cccc(-c2cc(-c3ccc(N4CCNCC4)cc3)on2)c1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 12/20 0.66
MAPKAPK2 P49137 3/20 0.51
PRKD3 O94806 1/20 0.49
PRKD2 Q9BZL6 1/20 0.49
BMPR1B O00238 1/20 0.47
ACVRL1 P37023 1/20 0.47
ACVR1 Q04771 1/20 0.47
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HTT P42858 1/20 0.45
MLLT1 Q03111 1/20 0.43
CTSK P43235 1/20 0.43
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6923596 0.90 PRKD1 (0.68) PRKD1PRKD3PRKD2NPC1RAB9A
SCHEMBL957994 0.89 PRKD1 (0.81) PRKD1PRKD3PRKD2ALDH1A1
SCHEMBL958900 0.86 PRKD1 (0.77) PRKD1PRKD3PRKD2ALDH1A1MLLT1
SCHEMBL6923075 0.84 PRKD1 (0.63) PRKD1PRKD3PRKD2SMN1; SMN2ALDH1A1
SCHEMBL6922372 0.82 PRKD1 (0.70) PRKD1PRKD3PRKD2ALDH1A1MLLT1
SCHEMBL937644 0.81 NPC1 (0.67) PRKD1PRKD3PRKD2NPC1RAB9A
SCHEMBL6923851 0.81 PRKD1 (0.63) PRKD1PRKD3PRKD2NPC1RAB9A
SCHEMBL959487 0.80 PRKD1 (0.76) PRKD1PRKD3PRKD2
SCHEMBL959488 0.80 PRKD1 (0.76) PRKD1PRKD3PRKD2
SCHEMBL966138 0.80 PRKD1 (0.62) PRKD1PRKD3PRKD2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009484-A1 ARYLPYRAZOLES AND ARYLISOXAZOLES AND THEIR USE AS PKD MODULATORS NOVARTIS AG (CH) 2011-01-27 WO disclosed