SCHEMBL9645251

SCHEMBL9645251

O=C1CCCN(c2ccccc2)N1C(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
HPGD P15428 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP2D6 P10635 1/20 0.50
NPC1 O15118 5/20 0.45
RAB9A P51151 5/20 0.45
KMT2A Q03164 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 2/20 0.45
TSHR P16473 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
F2 P00734 1/20 0.43
POLB P06746 2/20 0.43
HSD17B10 Q99714 1/20 0.43
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8590170 0.90 KMT2A (0.45) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
SCHEMBL9645410 0.79 MEN1 (0.43) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
SCHEMBL9645470 0.79 POLB (0.42) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
SCHEMBL1002469 0.75 CYP1A2 (0.64) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
SCHEMBL10417057 0.74 SMN1; SMN2 (0.45) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10417047 0.74 NAAA (0.49) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
Water SCHEMBL27387795 0.73 CYP1A2 (0.62) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
SCHEMBL11280055 0.72 KMT2A (0.37) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
SCHEMBL5674146 0.72 ALDH1A1 (0.45) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL11576464 0.71 NPC1 (0.51) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5086052-A Antiarthritic, antiallergens, antiinflammatory agents; also for asthma and psoriasis ABBOTT LABORATORIES (US) 1992-02-04 US disclosed
US-4970210-A ENZYME INHIBITORS ABBOTT LABORATORIES (US) 1990-11-13 US disclosed
EP-0299449-A2 Pyridazinone, triazinone and oxapyridazinone lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1989-01-18 EP disclosed