SCHEMBL9646646

SCHEMBL9646646

Fc1ccc(-c2[c]cccc2Br)cc1

nearest known ligand 0.32

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
MAPK13 O15264 1/20 0.31
GCGR P47871 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11705130 0.81 ALDH1A1 (0.44) L3MBTL1ALDH1A1TP53
SCHEMBL9265689 0.80 CYP1A2 (0.38) GRM2KDM4ECYP1A2HTTPTGS1
SCHEMBL150096 0.79 MAOB (0.32)
SCHEMBL5014600 0.78 PTGS2 (0.39) PTGS1PTGS2GCGRMAPK14ALDH1A1
SCHEMBL2012242 0.76 MAPK1 (0.38) HTTPTGS1PTGS2LMNATP53
SCHEMBL6131965 0.76 CYP3A4 (0.35) KDM4ECYP1A2CYP3A4HPGDCYP2C19
SCHEMBL9321438 0.76 PTGS2 (0.38) KDM4ECYP1A2CYP3A4HPGDCYP2C19
SCHEMBL2011907 0.76 KDM4E (0.38) KDM4ENPSR1PTGS1PTGS2MAPK14
SCHEMBL9650164 0.76 NPC1 (0.35) KDM4ECYP3A4HPGDHTTNPSR1
SCHEMBL9649234 0.74 ALDH1A1 (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120848-A Anticholesterol and antilipemic agents; hydroxy-3-methylglutaryl/3-/ coenzyme A reductase inhibitors GLAXO GROUP LIMITED (GB) 1992-06-09 US disclosed
US-5013749-A Imidazole derivatives and their use as hypercholesterolemia and hyperlipoproteinemia agents GLAXO GROUP LIMITED (GB) 1991-05-07 US disclosed