SCHEMBL9649697

SCHEMBL9649697

NCC(=O)Oc1ccc(O)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.42
CA1 P00915 2/20 0.41
NR1H4 Q96RI1 3/20 0.40
HSD17B10 Q99714 2/20 0.39
TSHR P16473 1/20 0.39
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
BACE1 P56817 1/20 0.36
ESR2 Q92731 2/20 0.35
ESR1 P03372 1/20 0.35
KDM4E B2RXH2 1/20 0.35
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10695957 0.86 KDM4E (0.43) CA2CA1TSHRHSP90AA1KDM4E
SCHEMBL10814685 0.84 MAPT (0.38) CA2CA1HSD17B10TSHRKDM4E
SCHEMBL11471018 0.83 KMT2A (0.50) CA2CA1NR1H4HSD17B10TSHR
SCHEMBL28642071 0.81 SOS1 (0.45) HSD17B10TSHRMAPTHTTKMT2A
SCHEMBL11528338 0.81 NPC1 (0.49) CA2ALDH1A1LMNAMAPTKMT2A
SCHEMBL17242255 0.80 MEN1 (0.53) CA2CA1NR1H4HSD17B10TSHR
SCHEMBL7391312 0.80 BCL9 (0.49) CA2CA1HSD17B10HSP90AA1HSP90AB1
SCHEMBL4789760 0.79 MAPT (0.38) NR1H4HSD17B10ESR2ESR1KDM4E
SCHEMBL28964153 0.78 ALDH1A1 (0.49) CA2CA1HSD17B10KDM4ETHRB
SCHEMBL4791444 0.77 TSHR (0.50) CA2CA1HSD17B10TSHRHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0494733-A1 Trifluoromethyl 1-carba(1-dethia)cephems ELI LILLY AND COMPANY (US) 1992-07-15 EP disclosed
US-5099015-A Antibiotics formed by bromination of trifluoromethanesulfonyl containing cephalosporins ELI LILLY AND COMPANY (US) 1992-03-24 US disclosed