SCHEMBL10695957

SCHEMBL10695957

NCC(=O)Oc1ccc(Cl)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 3/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
LMNA P02545 1/20 0.43
KMO O15229 2/20 0.42
CHRNA3 P32297 1/20 0.42
HSP90AA1 P07900 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP3A5 P20815 1/20 0.42
CYP2C19 P33261 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
HTR2A P28223 2/20 0.39
SLC6A4 P31645 2/20 0.39
KCNH2 Q12809 1/20 0.39
TSHR P16473 2/20 0.38
CA12 O43570 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9649697 0.86 CA2 (0.42) KDM4EALDH1A1LMNAHSP90AA1TSHR
SCHEMBL28642071 0.84 SOS1 (0.45) SMN1; SMN2HTR2ASLC6A4KCNH2TSHR
SCHEMBL1512534 0.81 ESR1 (0.53) KDM4EALDH1A1PPARGPPARALMNA
SCHEMBL27697768 0.81 KDM4E (0.43) KDM4EALDH1A1PPARGPPARALMNA
SCHEMBL3017398 0.79 BCL9 (0.51) KDM4EALDH1A1PPARGPPARALMNA
SCHEMBL2927179 0.79 KMT2A (0.47) KDM4EALDH1A1LMNASMN1; SMN2CA1
SCHEMBL23753577 0.79 MEN1 (0.57) KDM4EALDH1A1PPARGPPARALMNA
SCHEMBL28306740 0.77 KMT2A (0.46) KDM4EALDH1A1LMNACYP2D6CYP2C19
SCHEMBL28847251 0.77 KMT2A (0.46) KDM4EALDH1A1LMNACYP2D6CYP2C19
SCHEMBL19331388 0.76 WDR5 (0.47) KDM4EPPARGSMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101600700-B Novel 2-amino oxazolines as TAAR1 ligands for CNS disorders HOFFMANN LA ROCHE 2013-08-21 CN disclosed
CN-101600700-A Novel 2-aminooxazolines as TAAR1 ligands for CNS disorders HOFFMANN LA ROCHE (CH) 2009-12-09 CN disclosed
EP-0254578-A1 Antibiotic intermediates ELI LILLY AND COMPANY (US) 1988-01-27 EP disclosed