SCHEMBL9650334

SCHEMBL9650334

C=CCC(CO)C(O)c1ccccc1C

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.37
ESR1 P03372 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35
CYP2C19 P33261 1/20 0.34
ACP3 P15309 1/20 0.33
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
IDO1 P14902 1/20 0.30
TDO2 P48775 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9647516 0.83 CYP3A4 (0.39) SLC6A2SLC6A4CYP3A4CYP2D6SLC6A3
SCHEMBL9650127 0.83 LMNA (0.43) GAAKDM4ECYP1A2SLC6A2SLC6A4
SCHEMBL9650911 0.82 CES2 (0.36) SLC6A2SLC6A4CYP3A4CYP2D6SLC6A3
SCHEMBL3246301 0.79 GAA (0.41) GAAESR1KDM4ECYP1A2SLC6A2
SCHEMBL15184714 0.79 GAA (0.41) GAAESR1KDM4ECYP1A2SLC6A2
SCHEMBL9650174 0.77 CYP2C19 (0.49) KDM4ESLC6A2SLC6A4CYP3A4CYP2D6
SCHEMBL9715173 0.74 KRAS (0.30)
SCHEMBL4637099 0.73 ESR1 (0.42) GAAESR1SLC6A2SLC6A4CYP3A4
SCHEMBL13993318 0.73 ESR1 (0.59) GAAESR1KDM4ECYP1A2SLC6A2
SCHEMBL8995483 0.72 ESR1 (0.41) GAAESR1SLC6A2SLC6A4CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166377-A Thromboxane A2 antagonist as coagulants or vasoconstrictors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-11-24 US disclosed
US-4745198-A CARDIOVASCULAR DISORDERS, BRONCHODILATOR AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-05-17 US disclosed
EP-0094239-B1 1,3-DIOXAN-5-YLALKENOIC ACIDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-07-15 EP disclosed
US-4567197-A THORMBOXANE A2 ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-01-28 US disclosed
EP-0094239-A2 1,3-Dioxan-5-ylalkenoic acids IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-11-16 EP disclosed