SCHEMBL9650425

SCHEMBL9650425

FC1=CC[CH]C(c2cccc(Br)c2)=C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
ALDH1A1 P00352 4/20 0.35
BIRC5 O15392 1/20 0.34
NPY5R Q15761 1/20 0.34
RAB9A P51151 3/20 0.33
NPC1 O15118 2/20 0.33
HPGD P15428 2/20 0.33
TP53 P04637 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
IDO1 P14902 1/20 0.33
METAP2 P50579 1/20 0.33
CYP1A2 P05177 1/20 0.33
GABRP O00591 2/20 0.32
GABRD O14764 2/20 0.32
GABRA1 P14867 2/20 0.32
GABRB1 P18505 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9650518 0.80 HTR2C (0.37) CHRNB4CHRNA3ALDH1A1NPY5RRAB9A
SCHEMBL16579554 0.71 NPC1 (0.30) RAB9ANPC1
SCHEMBL29546450 0.66 ALDH1A1 (0.52) CHRNB4CHRNA3ALDH1A1BIRC5RAB9A
SCHEMBL312091 0.66 ALDH1A1 (0.52) CHRNB4CHRNA3ALDH1A1BIRC5RAB9A
SCHEMBL191276 0.64 ALDH1A1 (0.50) CHRNB4CHRNA3ALDH1A1BIRC5RAB9A
SCHEMBL26301211 0.64 ALDH1A1 (0.50) CHRNB4CHRNA3ALDH1A1BIRC5RAB9A
Water SCHEMBL28248751 0.64 ALDH1A1 (0.50) CHRNB4CHRNA3ALDH1A1BIRC5RAB9A
SCHEMBL15624388 0.64 ALDH1A1 (0.50) CHRNB4CHRNA3ALDH1A1BIRC5RAB9A
SCHEMBL29398919 0.64 ALDH1A1 (0.50) CHRNB4CHRNA3ALDH1A1BIRC5RAB9A
SCHEMBL9292507 0.64 TAAR1 (0.54) BIRC5NPY5RRAB9ANPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120848-A Anticholesterol and antilipemic agents; hydroxy-3-methylglutaryl/3-/ coenzyme A reductase inhibitors GLAXO GROUP LIMITED (GB) 1992-06-09 US disclosed
US-5013749-A Imidazole derivatives and their use as hypercholesterolemia and hyperlipoproteinemia agents GLAXO GROUP LIMITED (GB) 1991-05-07 US disclosed