SCHEMBL9651269

SCHEMBL9651269

C=CCOC(=O)C(=NOC)C(=O)CCl

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
PTP4A3 O75365 1/20 0.31
PTP4A2 Q12974 1/20 0.31
PTP4A1 Q93096 1/20 0.31
CYP3A4 P08684 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9651265 1.00 TSHR (0.33) TSHRPTP4A3PTP4A2PTP4A1CYP3A4
SCHEMBL9651169 0.84 PTP4A3 (0.33) TSHRPTP4A3PTP4A2PTP4A1CYP3A4
SCHEMBL9651164 0.84 PTP4A3 (0.33) TSHRPTP4A3PTP4A2PTP4A1CYP3A4
SCHEMBL9175808 0.81 CYP3A4 (0.33) TSHRCYP3A4
SCHEMBL9175802 0.81 CYP3A4 (0.33) TSHRCYP3A4
SCHEMBL9648194 0.80 ABCB1 (0.36) TSHR
SCHEMBL8626482 0.80 ABCB1 (0.36) TSHR
SCHEMBL9649935 0.77 ALDH1A1 (0.30)
SCHEMBL9649932 0.77 ALDH1A1 (0.30)
Alcohol SCHEMBL28489742 0.77 ABCB1 (0.35) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0246603-B1 4-HALOGENO-2-OXYIMINO-3-OXOBUTYRIC ACIDS Takeda Chemical Industries, Ltd. (JP) 1992-12-30 EP disclosed
CN-1014408-B PREPARATION OF 4-HALOGENO-2-OXYIMINO-3-OXOBUTYRIC ACID TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1991-10-23 CN disclosed
US-4845257-A 4-halogeno-2-oxyimino-3-oxobutyric acids and derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-07-04 US disclosed
CN-87103668-A 4-halo-2-oximino-3-ketobutyric acid 1988-04-13 CN disclosed
EP-0246603-A2 4-Halogeno-2-Oxyimino-3-Oxobutyric acids Takeda Chemical Industries, Ltd. (JP) 1987-11-25 EP disclosed