SCHEMBL9652008

SCHEMBL9652008

O=C(Cc1ccc(Cl)c(Cl)c1)N1CCN(Cc2ccccc2)CC1CO

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 11/20 0.56
SIGMAR1 Q99720 4/20 0.54
NPC1 O15118 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
NFKB1 P19838 1/20 0.54
CYP2C19 P33261 1/20 0.54
OPRD1 P41143 1/20 0.54
HIF1A Q16665 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
OPRM1 P35372 1/20 0.53
BLM P54132 1/20 0.53
PMP22 Q01453 1/20 0.53
DRD4 P21917 1/20 0.53
SLC6A3 Q01959 1/20 0.53
TMEM97 Q5BJF2 1/20 0.53
HTT P42858 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14367939 0.88 OPRK1 (0.73) OPRK1SIGMAR1NPC1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL5630292 0.87 OPRK1 (0.71) OPRK1SIGMAR1NPC1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL5630297 0.87 OPRK1 (0.71) OPRK1SIGMAR1NPC1CYP1A2CYP3A4
SCHEMBL9649179 0.85 OPRK1 (0.72) OPRK1NPC1CYP1A2CYP3A4CYP2D6
SCHEMBL9652026 0.84 OPRK1 (0.56) OPRK1SIGMAR1OPRD1OPRM1HTT
Fumaric Acid SCHEMBL9650695 0.84 BLM (0.70) OPRK1SIGMAR1NPC1CYP1A2CYP3A4
Maleic Acid SCHEMBL9650688 0.84 BLM (0.70) OPRK1SIGMAR1NPC1CYP1A2CYP3A4
SCHEMBL10416432 0.83 OPRK1 (0.62) OPRK1NPC1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7170793 0.82 OPRK1 (0.52) OPRK1SIGMAR1NPC1CYP1A2CYP3A4
SCHEMBL20528042 0.81 SIGMAR1 (0.51) SIGMAR1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116842-A Analgesics GLAXO GROUP LIMITED (GB) 1992-05-26 US disclosed
EP-0398720-A2 Piperazine derivatives GLAXO GROUP LIMITED (GB) 1990-11-22 EP disclosed
US-4943578-A ANALGESICS; CEREBRAL ANTIISCHEMIC AGENTS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed
EP-0343900-A2 Piperazine compounds GLAXO GROUP LIMITED (GB) 1989-11-29 EP disclosed