SCHEMBL9655394

SCHEMBL9655394

Cc1cc(C)nc(NC(=O)CC2(C)CCc3c(C)c(O)c(C)c(C)c3O2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.44
TSHR P16473 2/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
CYP1A2 P05177 1/20 0.44
USP2 O75604 2/20 0.44
CYP2C9 P11712 2/20 0.44
TP53 P04637 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
THPO P40225 1/20 0.44
HIF1A Q16665 1/20 0.44
LCK P06239 1/20 0.44
FYN P06241 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
DRD2 P14416 1/20 0.44
ADRA1D P25100 1/20 0.44
MAPK3 P27361 1/20 0.44
HTR2C P28335 1/20 0.44
MC4R P32245 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9655667 0.87 KMT2A (0.48) CYP3A4CYP1A2ALOX5KMT2AMEN1
SCHEMBL9313724 0.85 CYP3A4 (0.47) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9655147 0.85 PSEN1 (0.49) CYP3A4CYP1A2KMT2AMEN1MAPK1
SCHEMBL9313627 0.85 MEN1 (0.39) CYP3A4CYP1A2ALOX5LMNAKMT2A
SCHEMBL9314952 0.85 PSEN1 (0.38) CYP3A4CYP1A2MAPTKMT2ATDP1
SCHEMBL9428539 0.83 USP2 (0.46) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9427829 0.83 PTGS1 (0.56) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9313487 0.83 PSEN1 (0.40) CYP3A4CYP1A2LMNAKMT2AMEN1
SCHEMBL9314041 0.83 PSEN1 (0.42) CYP3A4CYP1A2KMT2AMEN1MAPK1
SCHEMBL9313502 0.82 BCHE (0.52) CYP3A4TSHRPTGS1PTGS2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512899-A1 Benzopyran compounds, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-11-11 EP disclosed