SCHEMBL9655419

SCHEMBL9655419

CCCCOC(=O)N[C@H]1CCN(OCc2ccccc2)C1=O

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 7/20 0.45
ALDH1A1 P00352 2/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CASP3 P42574 1/20 0.42
ASAH1 Q13510 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15382467 0.92 NAAA (0.47) NAAAALDH1A1CYP3A4TSHRMAPK1
SCHEMBL13244921 0.88 ALDH1A1 (0.51) NAAAALDH1A1TSHRCASP3
SCHEMBL18712231 0.88 ALDH1A1 (0.51) NAAAALDH1A1TSHRCASP3
SCHEMBL7842024 0.81 PREP (0.42) ALDH1A1
SCHEMBL9655228 0.81 KMT2A (0.48) L3MBTL1
SCHEMBL9655226 0.81 KMT2A (0.48) L3MBTL1
SCHEMBL4700151 0.77 ALDH1A1 (0.40) ALDH1A1
SCHEMBL10437936 0.77 ALDH1A1 (0.44) NAAAALDH1A1CYP3A4TSHRMAPK1
SCHEMBL4698575 0.76 ALDH1A1 (0.44) ALDH1A1
SCHEMBL19027637 0.76 KMT2A (0.50) L3MBTL1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0318091-B1 RESOLVED AMINO PYRROLIDINE NEUROPROTECTIVE AGENTS MERCK SHARP & DOHME LTD. (GB) 1992-12-09 EP disclosed
US-4863953-A [3R]-3-amino-1-hydroxy pyrrolidin-2-one and its use as a neuroprotective agent MERCK & CO., INC. (US) 1989-09-05 US disclosed
EP-0318091-A2 Resolved amino pyrrolidine neuroprotective agents MERCK SHARP & DOHME LTD. (GB) 1989-05-31 EP disclosed