SCHEMBL9656156

SCHEMBL9656156

COc1cc(CCN(C)CCCOc2ccc(S(=O)(=O)c3c(C(C)C)cn4ccccc34)cc2)cc(OC)c1

nearest known ligand 0.81

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAOB P27338 6/20 0.39
KCNH2 Q12809 2/20 0.38
SMPD1 P17405 4/20 0.38
MAOA P21397 2/20 0.36
LTA4H P09960 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9157509 0.91 CYP3A4 (0.50) KDM4ETP53CYP3A4MAPTTSHR
Hydrochloric Acid SCHEMBL9655914 0.91 CYP3A4 (0.49) KDM4ETP53CYP3A4MAPTTSHR
Fantofarone SCHEMBL29802340 0.90 CYP3A4 (0.59) KDM4ETP53CYP3A4MAPTTSHR
Fantofarone SCHEMBL77818 0.90 CYP3A4 (0.59) KDM4ETP53CYP3A4MAPTTSHR
Fantofarone SCHEMBL9599714 0.89 CYP3A4 (0.59) KDM4ETP53CYP3A4MAPTTSHR
SCHEMBL9215666 0.89 KDM4E (0.48) KDM4ETP53CYP3A4MAPTTSHR
SCHEMBL9152939 0.88 KDM4E (0.44) KDM4ETP53CYP3A4MAPTTSHR
SCHEMBL9598076 0.87 CYP3A4 (0.57) KDM4ETP53CYP3A4MAPTTSHR
SCHEMBL9272756 0.86 MEN1 (0.43) KDM4E
SCHEMBL9598438 0.84 CACNA1B (0.43) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5147878-A Hypotensive, antiarrhythmia agents SANOFI (FR) 1992-09-15 US claimed
US-5147878-A Hypotensive, antiarrhythmia agents SANOFI (FR) 1992-09-15 US disclosed