SCHEMBL9657693

SCHEMBL9657693

COP(=O)(C#Cc1c(-c2ccc(F)cc2)c(-c2ccccc2)n(C(C)C)c1C(C)C)C[C@@H](O)CC(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 5/20 0.44
ABCB11 O95342 2/20 0.44
NR1I2 O75469 1/20 0.44
RHOC P08134 1/20 0.44
CYP3A4 P08684 1/20 0.44
THRB P10828 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
SLCO1B1 Q9Y6L6 1/20 0.44
CYP2C9 P11712 3/20 0.41
SIRT6 Q8N6T7 2/20 0.41
ABCC3 O15438 1/20 0.41
PGR P06401 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
RXRA P19793 1/20 0.41
TBXA2R P21731 1/20 0.41
CCKAR P32238 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9516811 0.90 HMGCR (0.47) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9516800 0.90 HMGCR (0.47) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9655519 0.84 HMGCR (0.35) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9695065 0.83 ABCB11 (0.39) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9695052 0.83 ABCB11 (0.39) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL8953082 0.80
SCHEMBL9657698 0.79 HMGCR (0.43) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL8952710 0.79
SCHEMBL9657705 0.79 HMGCR (0.43) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL8953094 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0463456-A1 Phosphorus-containing HMG-CoA reductase inhibitors, new intermediates and their use E.R. SQUIBB & SONS, INC. (US) 1992-01-02 EP disclosed