SCHEMBL9665141

SCHEMBL9665141

COc1ccc(CCC(=O)C2CCCCC2=O)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.64
ALDH1A1 P00352 4/20 0.50
KMT2A Q03164 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
CYP2C19 P33261 1/20 0.50
F2RL1 P55085 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
EPHX2 P34913 1/20 0.46
KDM4E B2RXH2 1/20 0.45
TRPM8 Q7Z2W7 1/20 0.45
POLB P06746 1/20 0.45
FFAR1 O14842 1/20 0.45
FKBP1A P62942 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9663109 0.86 MAPK1 (0.51) MAPK1ALDH1A1POLBFKBP1A
SCHEMBL9662545 0.82 MCL1 (0.45) MAPK1ALDH1A1HPGDPOLB
SCHEMBL11728918 0.81 F2RL1 (0.57) MAPK1ALDH1A1KMT2ACYP1A2CYP3A4
SCHEMBL26637816 0.80 ALDH1A1 (0.60) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL7920767 0.79 MAPK1 (1.00) MAPK1ALDH1A1KMT2ACYP1A2CYP2D6
SCHEMBL7638791 0.76 KMT2A (0.47) MAPK1ALDH1A1KMT2ACYP1A2CYP2C9
SCHEMBL9663967 0.76 MCL1 (0.43) MAPK1KMT2APOLB
SCHEMBL535049 0.73 MCL1 (0.46) MAPK1ALDH1A1KMT2ACYP2D6HPGD
SCHEMBL5270856 0.73 MAPK1 (0.73) MAPK1ALDH1A1KMT2AHPGDPOLB
SCHEMBL10191436 0.73 ALDH1A1 (0.57) MAPK1ALDH1A1CYP1A2CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273451-B1 LIPOXYGENASE INHIBITORY COMPOUNDS Bristol-Myers Squibb Company (US) 1992-04-01 EP disclosed
US-4861798-A Lipoxygenase inhibitory compounds BRISTOL-MYERS COMPANY (US) 1989-08-29 US disclosed