SCHEMBL9665152

SCHEMBL9665152

CC(C)(C)OC(=O)CNC(=O)C(Cc1cccc2ccccc12)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.56
CTSK P43235 1/20 0.56
CTNNB1 P35222 1/20 0.50
CYP3A4 P08684 5/20 0.45
MME P08473 1/20 0.45
ACE P12821 1/20 0.45
CPA1 P15085 1/20 0.45
ACE2 Q9BYF1 1/20 0.45
HRH4 Q9H3N8 1/20 0.43
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
MMP14 P50281 1/20 0.41
VNN1 O95497 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27563011 0.87 CTSS (0.57) CTSSCTSKCTNNB1CYP3A4MME
SCHEMBL6318009 0.87 CTSS (0.57) CTSSCTSKCTNNB1CYP3A4MME
SCHEMBL9740320 0.79 CTSS (0.51) CTSSCTSKCTNNB1CYP3A4MME
SCHEMBL9668155 0.78 CTNNB1 (0.52) CTSSCTSKCTNNB1MMEACE
SCHEMBL10389693 0.78 CTNNB1 (0.52) CTSSCTSKCTNNB1MMEACE
SCHEMBL9668142 0.78 CTNNB1 (0.52) CTSSCTSKCTNNB1MMEACE
SCHEMBL9665156 0.77 CTNNB1 (0.51) CTSSCTSKCTNNB1CYP3A4MME
SCHEMBL613640 0.77 CTSS (0.76) CTSSCTSKCYP3A4MMEACE
SCHEMBL4600435 0.77 CTSS (0.76) CTSSCTSKCYP3A4MMEACE
SCHEMBL4122289 0.77 CTSS (0.76) CTSSCTSKCYP3A4MMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0184550-B1 5-AMINO-4-HYDROXY VALERYL AMIDE DERIVATIVES CIBA-GEIGY AG (CH) 1992-03-18 EP disclosed
US-4931591-A Novel 5-amino-4-hydroxyvaleryl derivatives CIBA-GEIGY CORPORATION (US) 1990-06-05 US disclosed
US-4727060-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1988-02-23 US disclosed
EP-0184550-A2 5-Amino-4-hydroxy valeryl amide derivatives CIBA-GEIGY AG (CH) 1986-06-11 EP disclosed