SCHEMBL9667403

SCHEMBL9667403

Cn1c(-c2ccc3[nH]c(-c4ccncc4)cc3c2)n[nH]c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.43
PDE3A Q14432 3/20 0.43
MMP2 P08253 1/20 0.41
MMP13 P45452 1/20 0.41
MMP14 P50281 1/20 0.41
MAPK9 P45984 1/20 0.40
MAPK10 P53779 1/20 0.40
CHEK1 O14757 1/20 0.39
HSD17B10 Q99714 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
GFER P55789 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CLK1 P49759 2/20 0.37
CDC7 O00311 2/20 0.36
NAMPT P43490 1/20 0.36
CLK2 P49760 1/20 0.36
CLK3 P49761 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9670178 0.86 CYP19A1 (0.52) MMP2MMP13MMP14CHEK1CLK2
SCHEMBL9668918 0.84 KDM4E (0.36) CHEK1HSD17B10KDM4EMAPTHPGD
SCHEMBL9669151 0.81 KDM4E (0.43) MAPK9MAPK10HSD17B10KDM4EMAPT
SCHEMBL9119099 0.78 MAPK9 (0.50) PDE3BPDE3AMAPK9MAPK10CHEK1
SCHEMBL31317792 0.76 CLK1 (0.54) PDE3BPDE3AMMP2MMP13MMP14
SCHEMBL21812414 0.76 CLK1 (0.54) PDE3BPDE3AMMP2MMP13MMP14
SCHEMBL9669274 0.76 CHRNA7 (0.44) HSD17B10KDM4EMAPTHPGDTSHR
SCHEMBL10556977 0.76 CLK2 (0.41) PDE3BPDE3AMAPK9MAPK10CHEK1
SCHEMBL16382915 0.73 NPC1 (0.56) HSD17B10KDM4EMAPTHPGDGFER
SCHEMBL10553367 0.72 PDE3B (0.42) PDE3BPDE3AMMP2MMP13MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223937-B1 INDOLES SUBSTITUTED WITH HETEROCYCLES, INTERMEDIATES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS Roche Diagnostics GmbH (DE) 1992-03-18 EP disclosed