SCHEMBL9669151

SCHEMBL9669151

Cn1c(-c2ccc3[nH]c(-c4ccccn4)cc3c2)n[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ITK Q08881 4/20 0.40
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
CDK5 Q00535 2/20 0.39
CDK5R1 Q15078 2/20 0.39
METAP2 P50579 1/20 0.38
METAP1 P53582 1/20 0.38
CBFB Q13951 1/20 0.38
BTK Q06187 1/20 0.37
PDE10A Q9Y233 2/20 0.37
GCK P35557 2/20 0.36
NPY5R Q15761 1/20 0.36
CCNB2 O95067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9667403 0.81 PDE3B (0.43) KDM4EHPGDGSK3BMAPK9MAPK10
SCHEMBL9670178 0.80 CYP19A1 (0.52) ALDH1A1BTK
SCHEMBL9668918 0.76 KDM4E (0.36) KDM4EHPGDNPC1ALDH1A1LMNA
SCHEMBL28784366 0.75 ITK (0.57) KDM4EHPGDNPC1ALDH1A1LMNA
SCHEMBL9669274 0.72 CHRNA7 (0.44) KDM4EHPGDALDH1A1MAPTTSHR
SCHEMBL10554267 0.70 SMN1; SMN2 (0.47) KDM4EHPGDNPC1ALDH1A1LMNA
SCHEMBL308319 0.70 GSK3B (0.61) KDM4EHPGDNPC1ALDH1A1LMNA
SCHEMBL29470995 0.70 GSK3B (0.61) KDM4EHPGDNPC1ALDH1A1LMNA
SCHEMBL1466825 0.69 SMN1; SMN2 (0.55) KDM4EHPGDNPC1ALDH1A1LMNA
SCHEMBL31317744 0.68 CYP11B1 (0.50) KDM4ENPC1RAB9ASMN1; SMN2ITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223937-B1 INDOLES SUBSTITUTED WITH HETEROCYCLES, INTERMEDIATES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS Roche Diagnostics GmbH (DE) 1992-03-18 EP disclosed
US-4851406-A CARDIOVASCULAR DISORDERS, HYPOTENSIVE BOEHRINGER MANNHEIM GMBH (DE) 1989-07-25 US disclosed