SCHEMBL9668355

SCHEMBL9668355

COc1cc2c(cc1OC)C(=O)NC(CCCCl)C2

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.44
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
PDE4D Q08499 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4858398 0.77 ACHE (0.56) ACHE
SCHEMBL4853298 0.73 ACHE (0.55) ACHE
SCHEMBL10519759 0.71 ACHE (0.44) ACHE
Hydrochloric Acid SCHEMBL10521614 0.71 ACHE (0.43) ACHE
SCHEMBL12043675 0.71 ACHE (0.50) ACHEKDM4EALDH1A1KMT2A
SCHEMBL10854754 0.70 ACHE (0.49) ACHEKDM4EALDH1A1KMT2A
SCHEMBL10645687 0.67 MAOA (0.45) ACHEALDH1A1KMT2A
SCHEMBL10848767 0.64 SRC (0.40) KMT2A
SCHEMBL10200127 0.64 CYP3A4 (0.49) ACHEKDM4EALDH1A1KMT2A
SCHEMBL10656149 0.63 GRM2 (0.45) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0259793-B1 NAPHTHYL DERIVATIVES, MEDICAMENTS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1992-07-01 EP disclosed
US-4871735-A HYPOTENSIVE, ANTIISCHEMIC AGENTS DR. KARL THOMAE GMBH 1989-10-03 US disclosed
EP-0259793-A1 Naphthyl derivatives, medicaments containing them and processes for their preparation Dr. Karl Thomae GmbH (DE) 1988-03-16 EP disclosed