SCHEMBL9668644

SCHEMBL9668644

O=C1C=CC(Cl)(C(=O)OCc2ccccc2)O1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
DDB1 Q16531 1/20 0.43
CRBN Q96SW2 1/20 0.43
TDP1 Q9NUW8 2/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KMT2A Q03164 1/20 0.41
MGLL Q99685 1/20 0.39
CDC25B P30305 1/20 0.39
LMNA P02545 1/20 0.39
HCAR2 Q8TDS4 1/20 0.39
TSHR P16473 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4609023 0.70 DDB1 (0.54) ALDH1A1DDB1CRBNTDP1MAPK1
SCHEMBL4607575 0.70 ALDH1A1 (0.45) ALDH1A1DDB1CRBNTDP1MAPK1
SCHEMBL10726489 0.69 ALDH1A1 (0.55) ALDH1A1DDB1CRBNTDP1MAPK1
SCHEMBL15095465 0.68 ALDH1A1 (0.58) ALDH1A1DDB1CRBNTDP1MAPK1
SCHEMBL4272254 0.68 DDB1 (0.51) ALDH1A1DDB1CRBNTDP1MAPK1
SCHEMBL21160844 0.67 CTRB1 (0.45) ALDH1A1DDB1CRBNTDP1MAPK1
SCHEMBL16661304 0.66 DDB1 (0.56) ALDH1A1DDB1CRBNTDP1MAPK1
SCHEMBL20156647 0.66 DDB1 (0.46) ALDH1A1DDB1CRBNTDP1MAPK1
Hydrazine SCHEMBL28257347 0.66 ALDH1A1 (0.92) ALDH1A1TDP1MAPK1L3MBTL1SLC6A2
SCHEMBL1504008 0.65 DDB1 (0.59) ALDH1A1DDB1CRBNTDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0219923-B1 ANTIBIOTIC DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-09-02 EP claimed
EP-0219923-B1 ANTIBIOTIC DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1992-09-02 EP disclosed
US-4851422-A Antibiotic 2-(3-oxo-2-isoxazolidinyl)-5-oxo-2-tetrahydrofuran-carboxylates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-07-25 US disclosed
EP-0219923-A1 Antibiotic derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-04-29 EP disclosed