SCHEMBL9670280

SCHEMBL9670280

CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccccc1N

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 6/20 0.52
CTSS P25774 1/20 0.50
CTSK P43235 1/20 0.50
CA2 P00918 1/20 0.49
HDAC1 Q13547 1/20 0.46
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
GLS O94925 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ATM Q13315 1/20 0.44
TRPA1 O75762 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4080775 0.91 AAK1 (0.51) AAK1CTSSCTSKCA2HDAC1
SCHEMBL9744622 0.88 CTSS (0.55) AAK1CTSSCTSKCA2HDAC1
SCHEMBL9286086 0.87 AAK1 (0.51) AAK1CTSSCTSKHDAC1LMNA
SCHEMBL9283981 0.87 AAK1 (0.51) AAK1CTSSCTSKHDAC1LMNA
SCHEMBL8345117 0.86 CTSS (0.51) CTSSCTSKCA2LMNAPOLB
SCHEMBL8347951 0.86 CTSS (0.51) CTSSCTSKCA2LMNAPOLB
SCHEMBL8344155 0.86 CTSS (0.51) CTSSCTSKCA2LMNAPOLB
SCHEMBL5349230 0.83 HDAC1 (0.48) AAK1CTSSCTSKHDAC1MEN1
SCHEMBL29412673 0.83 SMN1; SMN2 (0.52) AAK1CTSSCTSKCA2GLS
SCHEMBL29156938 0.83 SMN1; SMN2 (0.52) AAK1CTSSCTSKCA2GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0485458-A1 THIOACYLATING REAGENTS AND INTERMEDIATES, THIOPEPTIDES, AND METHODS FOR PREPARING AND USING SAME. IAF BIOCHEM INT (CA) 1992-05-20 EP claimed
WO-1991001976-A1 THIOACYLATING REAGENTS AND INTERMEDIATES, THIOPEPTIDES, AND METHODS FOR PREPARING AND USING SAME IAF BIOCHEM INTERNATIONAL INC. (CA) 1991-02-21 WO claimed