SCHEMBL9675375

SCHEMBL9675375

O=C1CCn2c(CO)nc3cccc1c32

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.45
HTR3A P46098 1/20 0.41
KCNH2 Q12809 4/20 0.39
GRM2 Q14416 4/20 0.39
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
PABPC1 P11940 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8483043 0.81 PARP1 (0.69) PARP1HTR3AKCNH2GRM2MAPT
SCHEMBL6139222 0.78 PARP1 (0.44) PARP1HTR3AKCNH2GRM2MAPT
Ethylene SCHEMBL6511634 0.75 PARP1 (0.42) PARP1HTR3AKCNH2GRM2MAPT
SCHEMBL6199833 0.74 PARP1 (0.66) PARP1HTR3AKCNH2GRM2
SCHEMBL7257414 0.73 KCNH2 (0.39) PARP1HTR3AKCNH2GRM2
SCHEMBL7265551 0.72 ATM (0.45) PARP1HTR3AKCNH2GRM2
SCHEMBL7257136 0.72 OPRM1 (0.37) PARP1HTR3AKCNH2GRM2
SCHEMBL6630805 0.71 PARP1 (0.43) PARP1HTR3A
SCHEMBL8824023 0.71 PARP1 (0.68) PARP1HTR3AKCNH2GRM2
SCHEMBL7257413 0.71 PARP1 (0.36) PARP1HTR3AKCNH2GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276942-B1 6-BETA(SUBSTITUTED)-(S)-HYDROXYMETHYLPENICILLANIC ACIDS AND DERIVATIVES THEREOF PFIZER INC. (US) 1992-04-01 EP disclosed
US-4782050-A BACTERICIDES PFIZER INC. (US) 1988-11-01 US disclosed
EP-0276942-A1 6-Beta(substituted)-(S)-hydroxymethylpenicillanic acids and derivatives thereof PFIZER INC. (US) 1988-08-03 EP disclosed