SCHEMBL9680146

SCHEMBL9680146

c1ccc2c(c1)CC(N1CCN(c3nsc4ccccc34)CC1)C2

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
MAPT P10636 1/20 0.56
HTR1A P08908 1/20 0.49
DRD2 P14416 1/20 0.49
HTR2A P28223 1/20 0.49
DRD3 P35462 1/20 0.49
SORD Q00796 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10843856 0.91 KDM4E (0.50) KDM4EMAPTHTR1ADRD2HTR2A
SCHEMBL10848984 0.84 KDM4E (0.57) KDM4EMAPTHTR1ADRD2HTR2A
SCHEMBL7777530 0.83 KDM4E (0.56) KDM4EMAPTHTR1ADRD2HTR2A
SCHEMBL9722202 0.81 DRD2 (0.59) KDM4EMAPTHTR1ADRD2HTR2A
SCHEMBL6884485 0.79 KDM4E (0.65) KDM4EMAPTHTR1ADRD2HTR2A
SCHEMBL5090039 0.79 KDM4E (0.54) KDM4EMAPTHTR1ADRD2HTR2A
Hydrochloric Acid SCHEMBL8401502 0.78 KDM4E (0.68) KDM4EMAPTHTR1ADRD2HTR2A
SCHEMBL4558892 0.77 KDM4E (0.71) KDM4EMAPTHTR1ADRD2HTR2A
SCHEMBL9381820 0.77 HTR1A (0.48) HTR1ADRD2HTR2A
SCHEMBL11637734 0.76 KDM4E (0.65) KDM4EMAPTHTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4590196-A NON-OPIATE BRISTOL-MYERS COMPANY (US) 1986-05-20 US claimed
US-5173490-A Antipsychotic drugs having no side effects; anxiolytic agents; analgesics; tranquilizers; sedatives; antidepressants ADIR ET COMPAGNIE (FR) 1992-12-22 US disclosed
EP-0494817-A1 Benzisoxazole and benzisothiazole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-07-15 EP disclosed