SCHEMBL9680680

SCHEMBL9680680

CN1CCN(c2nn(-c3ccc(O)cc3)c3ccccc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KHK P50053 2/20 0.48
SOS2 Q07890 1/20 0.47
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
RAD52 P43351 1/20 0.46
HTR3E A5X5Y0 2/20 0.43
HTR3B O95264 2/20 0.43
HTR3A P46098 2/20 0.43
HTR3D Q70Z44 2/20 0.43
HTR3C Q8WXA8 2/20 0.43
HRH4 Q9H3N8 3/20 0.43
PTGER1 P34995 2/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ESR2 Q92731 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6125292 0.89 KHK (0.56) KHKHTR3EHTR3BHTR3AHTR3D
SCHEMBL9762766 0.88 KHK (0.52) KHKMAPTHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9682152 0.87 KHK (0.54) KHKHTR3EHTR3BHTR3AHTR3D
SCHEMBL9681940 0.86 KHK (0.48) KHKLMNAHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9681492 0.86 KHK (0.51) KHKMAPTHTR3EHTR3BHTR3A
SCHEMBL9681274 0.84 HRH4 (0.49) KHKLMNAGAAMAPTHRH4
SCHEMBL9681720 0.84 KHK (0.47) KHKMAPTHTR3EHTR3BHTR3A
SCHEMBL9680624 0.83 CYP1A2 (0.46) KHKLMNAMAPTHTR3EHTR3B
Hydrochloric Acid SCHEMBL9680640 0.83 HRH4 (0.48) KHKLMNAGAAMAPTHRH4
SCHEMBL9763071 0.82 PTGER1 (0.44) LMNAGAAMAPTPTGER1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed