SCHEMBL9763071

SCHEMBL9763071

NC(=O)N1CCN(c2nn(-c3ccc(O)cc3)c3ccccc23)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 2/20 0.44
ME2 P23368 5/20 0.42
ME1 P48163 5/20 0.42
ME3 Q16798 5/20 0.42
SCN9A Q15858 1/20 0.42
MGLL Q99685 2/20 0.41
HTR1A P08908 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.39
HTR6 P50406 1/20 0.39
ALDH1A1 P00352 3/20 0.38
LMNA P02545 3/20 0.38
GAA P10253 3/20 0.38
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KIT P10721 1/20 0.38
USP2 O75604 1/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681935 0.91 PTGER1 (0.49) PTGER1SCN9AMGLLHTR1AHTR2A
SCHEMBL9680653 0.89 PTGER1 (0.43) PTGER1SCN9AALDH1A1LMNAMAPT
SCHEMBL9680606 0.89 TP53 (0.45) PTGER1SCN9ALMNAMAPTKIT
SCHEMBL9763297 0.86 SCN9A (0.46) PTGER1ME2ME1ME3SCN9A
SCHEMBL9682459 0.86 POLB (0.47) SCN9AMGLLLMNAGAAMAPT
SCHEMBL9680680 0.82 KHK (0.48) PTGER1LMNAGAAMAPTMEN1
SCHEMBL9681720 0.80 KHK (0.47) PTGER1HTR6MAPTESR2KDM4E
SCHEMBL9681280 0.80 LMNA (0.45) PTGER1SCN9AMGLLALDH1A1LMNA
SCHEMBL9680660 0.80 PTGER1 (0.43) PTGER1HTR1AHTR2AHTR7HTR6
SCHEMBL9681937 0.78 KHK (0.42) PTGER1HTR1AHTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed