SCHEMBL9681940

SCHEMBL9681940

CN1CCN(c2nn(-c3ccc(F)cc3)c3ccccc23)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 2/20 0.48
HTR6 P50406 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
HRH4 Q9H3N8 4/20 0.44
HTR3E A5X5Y0 2/20 0.43
HTR3B O95264 2/20 0.43
HTR3A P46098 2/20 0.43
HTR3D Q70Z44 2/20 0.43
HTR3C Q8WXA8 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTR1A P08908 1/20 0.41
HTR2C P28335 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9681228 0.90 LMNA (0.44) KHKHTR6CYP3A4CYP2D6MEN1
Fumaric Acid SCHEMBL9681236 0.90 LMNA (0.44) KHKHTR6CYP3A4CYP2D6MEN1
SCHEMBL6125292 0.89 KHK (0.56) KHKHTR6HRH4HTR3EHTR3B
SCHEMBL9762766 0.88 KHK (0.52) KHKHRH4HTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9682152 0.87 KHK (0.54) KHKHRH4HTR3EHTR3BHTR3A
SCHEMBL9682530 0.86 KHK (0.51) KHKHTR6HRH4HTR3EHTR3B
SCHEMBL9680680 0.86 KHK (0.48) KHKHRH4HTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9681492 0.86 KHK (0.51) KHKHRH4HTR3EHTR3BHTR3A
SCHEMBL9680624 0.86 CYP1A2 (0.46) KHKCYP3A4CYP2D6HRH4HTR3E
SCHEMBL9763064 0.86 KHK (0.51) KHKCYP3A4CYP2D6HRH4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
JP-1066171-A None JP disclosed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed