SCHEMBL9682489

SCHEMBL9682489

FC(F)(F)c1ccc(-n2nc(N3CCNCC3)c3ccccc32)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.47
HTR1D P28221 2/20 0.46
HTR2C P28335 2/20 0.46
KHK P50053 4/20 0.44
HTR3A P46098 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
MAPT P10636 2/20 0.43
THRB P10828 1/20 0.43
HTR1A P08908 1/20 0.43
RAB9A P51151 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP1A2 P05177 1/20 0.42
EPHX2 P34913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9680573 0.99 HTR6 (0.46) HTR6HTR1DHTR2CKHKHTR3A
SCHEMBL9681305 0.86 KHK (0.47) HTR6HTR2CKHKHTR3AMAPT
SCHEMBL9683199 0.85 HTR1D (0.51) HTR6HTR1DHTR2CKHKHTR3A
SCHEMBL2710715 0.85 KHK (0.54) HTR6HTR2CKHKHTR3AHTR3E
SCHEMBL9680624 0.85 CYP1A2 (0.46) HTR1DHTR2CKHKHTR3AHTR3E
Hydrochloric Acid SCHEMBL9681346 0.84 KHK (0.53) HTR6HTR2CKHKHTR3AHTR3E
SCHEMBL9681867 0.83 KHK (0.53) HTR2CKHKHTR3AADRB1
SCHEMBL9681720 0.83 KHK (0.47) HTR6HTR2CKHKHTR3AHTR3E
SCHEMBL9681327 0.83 KHK (0.47) HTR6HTR2CKHKMAPTKDM4E
Hydrochloric Acid SCHEMBL9680719 0.82 KHK (0.52) HTR2CKHKHTR3AMAPTHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed