SCHEMBL968136

SCHEMBL968136

C=CCc1cccc([O])c1CC=C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.47
GABRB2 P47870 2/20 0.47
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
MAPT P10636 2/20 0.38
MAPK1 P28482 1/20 0.38
AKR1B1 P15121 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 4/20 0.33
GAA P10253 3/20 0.33
LMNA P02545 3/20 0.33
ALOX12 P18054 2/20 0.33
POLB P06746 1/20 0.33
MTNR1A P48039 1/20 0.33
KDM4E B2RXH2 4/20 0.33
HSD17B10 Q99714 3/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18136 0.84 GABRA1 (0.56) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL9397812 0.81 GABRA1 (0.35) GABRA1GABRB2POLB
SCHEMBL384205 0.80 GABRA1 (0.47) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL4170461 0.78 GABRA1 (0.50) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL2362269 0.78 GABRA1 (0.61) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL4456728 0.78 GABRA1 (0.54) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL12076599 0.78 GABRA1 (0.54) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL8961782 0.78 MAPT (0.37) GABRA1GABRB2KMT2AMAPTL3MBTL1
SCHEMBL4863557 0.77 GABRA1 (0.48) GABRA1GABRB2KMT2AMEN1MAPT
SCHEMBL10625097 0.77 GABRA1 (0.48) GABRA1GABRB2KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547749-B2 Triazine compounds, polymers comprising triazine structural units, and method SABIC INNOVATIVE PLATICS IP B.V. (NL) 2009-06-16 US claimed
US-20080097040-A1 TRIAZINE COMPOUNDS, POLYMERS COMPRISING TRIAZINE STRUCTURAL UNITS, AND METHOD GENERAL ELECTRIC COMPANY (US) 2008-04-24 US claimed
US-20050192411-A1 Triazine compounds, polymers comprising triazine structural units, and method GENERAL ELECTRIC CO. 2005-09-01 US claimed
EP-1423372-A2 TRIAZINE COMPOUNDS, POLYMERS COMPRISING TRIAZINE STRUCTURAL UNITS, AND PROCESSES FOR THE PREPARATION OF THESE POLYMERS GENERAL ELECTRIC COMPANY (US) 2004-06-02 EP claimed
US-20030078347-A1 Triazine compounds, polymers comprising triazine structural units, and method GENERAL ELECTRIC COMPANY 2003-04-24 US claimed
WO-2003024939-A2 TRIAZINE COMPOUNDS POLYMERS COMPRISING TRIAZINE STRUCTURAL UNITS, AND PROCESSES FOR THE PREPARATION OF THESE POLYMERS GENERAL ELECTRIC COMPANY (US) 2003-03-27 WO claimed
US-5286266-A Motor fuel detergent additives - asymmetrical ureas of hydrocarbyloxypolyether amines and tertiary aminoalkyl primary amines TEXACO INC. (US) 1994-02-15 US claimed
EP-0403511-B1 HYDROGENATION OF HALONITROAROMATIC COMPOUNDS EASTMAN KODAK COMPANY (US) 1993-03-24 EP claimed
EP-0217485-B1 ACRYLIC-METHYLENE SUCCINIC ESTER EMULSION COPOLYMERS FOR THICKENING AQUEOUS SYSTEMS National Starch and Chemical Investment Holding Corporation (US) 1991-07-24 EP claimed
EP-0403511-A1 HYDROGENATION OF HALONITROAROMATIC COMPOUNDS. EASTMAN KODAK CO (US) 1990-12-27 EP claimed
US-4929737-A FORMING AMINOHALOAROMATIC COMPOUNDS EASTMAN KODAK COMPANY (US) 1990-05-29 US claimed
US-4877617-A COATING WITH SOLUTION OF QUATERNARY AMMONIUM SALT OF ALGINIC ACID OR CMC IN REMOVABLE SOLVENT; HOUSEHOLDS, MEDICINE, INDUSTRY DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1989-10-31 US claimed
WO-1989007096-A1 HYDROGENATION OF HALONITROAROMATIC COMPOUNDS EASTMAN KODAK COMPANY (US) 1989-08-10 WO claimed
US-4745154-A THICKENERS, FLOCCULANTS, DRILLING FLUIDS ALCO CHEMICAL CORPORATION (US) 1988-05-17 US claimed
EP-0217485-A2 Acrylic-methylene succinic ester emulsion copolymers for thickening aqueous systems National Starch and Chemical Investment Holding Corporation (US) 1987-04-08 EP claimed
EP-0197635-A2 Acrylic emulsion copolymers for thickening aqueous systems and copolymerizable surfactant monomers for use therein National Starch and Chemical Investment Holding Corporation (US) 1986-10-15 EP claimed
EP-0025775-B1 PROCESS FOR THE PRODUCTION OF A MONOCHROMATIC COLOUR IMAGE, AND PHOTOGRAPHIC MATERIAL SUITED THEREFOR CIBA-GEIGY AG (CH) 1985-05-29 EP claimed
US-4315069-A FORMING A MONOCHROMATIC DYE IMAGE CIBA GEIGY AG (CH) 1982-02-09 US claimed
US-4208345-A 2-Hydroxy-n-propylamine derivatives useful as surface active agents SANDOZ LTD. (CH) 1980-06-17 US claimed
JP-1207476-A None JP disclosed
EP-3888566-A1 SURGICAL STAPLER COMPRISING TISSUE THICKNESS COMPENSATORS Ethicon LLC (PR) 2021-10-06 EP disclosed
EP-2644122-B1 SURGICAL STAPLER COMPRISING TISSUE THICKNESS COMPENSATORS ETHICON LLC (PR) 2021-03-10 EP disclosed
WO-2019007922-A1 SOLID PIGMENT DISPERSION, PROCESS FOR PREPARING THE SAME AND PROCESS FOR PREPARING AQUEOUS OR ORGANIC SOLVENT-BASED INKJET INK CLARIANT INTERNATIONAL LTD (CH) 2019-01-10 WO disclosed
EP-1423372-B1 TRIAZINE COMPOUNDS, POLYMERS COMPRISING TRIAZINE STRUCTURAL UNITS, AND PROCESSES FOR THE PREPARATION OF THESE POLYMERS SABIC GLOBAL TECHNOLOGIES BV (NL) 2016-07-20 EP disclosed
US-8697811-B2 Curable resin composition and cured resin KURARAY CO., LTD. (JP) 2014-04-15 US disclosed
US-20130295349-A1 TRANSPARENT CONDUCTIVE FILM WITH PRESSURE-SENSITIVE ADHESIVE LAYER, METHOD FOR PRODUCING SAME, AND TOUCH PANEL NITTO DENKO CORPORATION (JP) 2013-11-07 US disclosed
WO-2013148789-A1 TISSUE THICKNESS COMPENSATORS ETHICON ENDO-SURGERY, INC. (US) 2013-10-03 WO disclosed
EP-2644122-A1 Tissue thickness compensators Ethicon Endo-Surgery, Inc. (US) 2013-10-02 EP disclosed
EP-2253666-B1 CURABLE RESIN COMPOSITION AND CURED RESIN KURARAY CO (JP) 2012-05-23 EP disclosed
US-20110003947-A1 CURABLE RESIN COMPOSITION AND CURED RESIN KURARAY CO., LTD. (JP) 2011-01-06 US disclosed
EP-2253666-A1 CURABLE RESIN COMPOSITION AND CURED RESIN Kuraray Co., Ltd. (JP) 2010-11-24 EP disclosed
US-7547749-B2 Triazine compounds, polymers comprising triazine structural units, and method SABIC INNOVATIVE PLATICS IP B.V. (NL) 2009-06-16 US disclosed
US-20080097040-A1 TRIAZINE COMPOUNDS, POLYMERS COMPRISING TRIAZINE STRUCTURAL UNITS, AND METHOD GENERAL ELECTRIC COMPANY (US) 2008-04-24 US disclosed
US-7235611-B2 Triazine compounds, polymers comprising triazine structural units, and method GENERAL ELECTRIC COMPANY (US) 2007-06-26 US disclosed
US-20050192411-A1 Triazine compounds, polymers comprising triazine structural units, and method GENERAL ELECTRIC CO. 2005-09-01 US disclosed
EP-1423372-A2 TRIAZINE COMPOUNDS, POLYMERS COMPRISING TRIAZINE STRUCTURAL UNITS, AND PROCESSES FOR THE PREPARATION OF THESE POLYMERS GENERAL ELECTRIC COMPANY (US) 2004-06-02 EP disclosed
US-20030078347-A1 Triazine compounds, polymers comprising triazine structural units, and method GENERAL ELECTRIC COMPANY 2003-04-24 US disclosed
WO-2003024939-A2 TRIAZINE COMPOUNDS POLYMERS COMPRISING TRIAZINE STRUCTURAL UNITS, AND PROCESSES FOR THE PREPARATION OF THESE POLYMERS GENERAL ELECTRIC COMPANY (US) 2003-03-27 WO disclosed
JP-2000160027-A ANTIBACTERIAL COMPOSITION DAICEL CHEM IND LTD 2000-06-13 JP disclosed
JP-2000026212-A ANTIMICROBIAL PARTICLE AND ITS PRODUCTION DAICEL CHEM IND LTD 2000-01-25 JP disclosed
EP-0453010-B1 Copolymer compositions comprising a copolymer and one or more lubricating additives SHELL INT RESEARCH (NL) 1996-06-05 EP disclosed
EP-0443685-B1 Process for the preparation of copolymers of carbon monoxide with one or more olefinically unsaturated compounds SHELL INT RESEARCH (NL) 1996-05-08 EP disclosed
EP-0315876-B1 Dispersion copolymers containing urethane groups, based on olefinically unsaturated monomers, process for their preparation and their use HOECHST AG (DE) 1996-04-10 EP disclosed
EP-0450695-B1 Copolymer compositions comprising a copolymer and one or more lubricating additives SHELL INT RESEARCH (NL) 1996-01-17 EP disclosed
US-5286266-A Motor fuel detergent additives - asymmetrical ureas of hydrocarbyloxypolyether amines and tertiary aminoalkyl primary amines TEXACO INC. (US) 1994-02-15 US disclosed
EP-0403511-B1 HYDROGENATION OF HALONITROAROMATIC COMPOUNDS EASTMAN KODAK COMPANY (US) 1993-03-24 EP disclosed
US-5115002-A Carbon monoxide-ethylene copolymer and a zeolite stabilizer SHELL OIL COMPANY (US) 1992-05-19 US disclosed
US-5093414-A Protective coatings for steels HOECHST AKTIENGESELLSCHAFT (DE) 1992-03-03 US disclosed
US-5075422-A PROCESS FOR THE PREPARATION OF POLYKETONE COPOLYMERS AND COPOLYMER WASH WITH LIQUID COMPRISING CARBOXYLIC COMPOUND SHELL OIL COMPANY (US) 1991-12-24 US disclosed
EP-0453010-A1 Copolymer compositions comprising a copolymer and one or more lubricating additives SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-10-23 EP disclosed
EP-0450695-A1 Copolymer compositions comprising a copolymer and one or more lubricating additives SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-10-09 EP disclosed
EP-0443685-A2 Process for the preparation of copolymers of carbon monoxide with one or more olefinically unsaturated compounds SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-08-28 EP disclosed
EP-0217485-B1 ACRYLIC-METHYLENE SUCCINIC ESTER EMULSION COPOLYMERS FOR THICKENING AQUEOUS SYSTEMS National Starch and Chemical Investment Holding Corporation (US) 1991-07-24 EP disclosed
EP-0403511-A1 HYDROGENATION OF HALONITROAROMATIC COMPOUNDS. EASTMAN KODAK CO (US) 1990-12-27 EP disclosed
US-4929737-A FORMING AMINOHALOAROMATIC COMPOUNDS EASTMAN KODAK COMPANY (US) 1990-05-29 US disclosed
US-4877617-A COATING WITH SOLUTION OF QUATERNARY AMMONIUM SALT OF ALGINIC ACID OR CMC IN REMOVABLE SOLVENT; HOUSEHOLDS, MEDICINE, INDUSTRY DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1989-10-31 US disclosed
JP-H01207476-A ANTIFUNGAL TREATMENT OF TEXTILES DAICEL CHEM IND LTD 1989-08-21 JP disclosed
WO-1989007096-A1 HYDROGENATION OF HALONITROAROMATIC COMPOUNDS EASTMAN KODAK COMPANY (US) 1989-08-10 WO disclosed
EP-0315876-A2 Dispersion copolymers containing urethane groups, based on olefinically unsaturated monomers, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1989-05-17 EP disclosed
US-4745154-A THICKENERS, FLOCCULANTS, DRILLING FLUIDS ALCO CHEMICAL CORPORATION (US) 1988-05-17 US disclosed
EP-0197635-A2 Acrylic emulsion copolymers for thickening aqueous systems and copolymerizable surfactant monomers for use therein National Starch and Chemical Investment Holding Corporation (US) 1986-10-15 EP disclosed
US-4419283-A AT LEAST THREE MUTUALLY IMMISCIBLE LIQUID PHASES SCHNEIDER RONALD A 1983-12-06 US disclosed
US-4208345-A 2-Hydroxy-n-propylamine derivatives useful as surface active agents SANDOZ LTD. (CH) 1980-06-17 US disclosed
US-4151149-A OXYGEN BARRIER MEMBRANES, SULFATED MONOMERS UNION OIL COMPANY OF CALIFORNIA (US) 1979-04-24 US disclosed
US-4044032-A LUBRICATING OILS TEXACO INC. (US) 1977-08-23 US disclosed
US-3944495-A AUTOMATIC TRANSMISSION FLUID TEXACO INC. (US) 1976-03-16 US disclosed
US-3944495-A AUTOMATIC TRANSMISSION FLUID TEXACO INC. (US) 1976-03-16 US disclosed