SCHEMBL9681660

SCHEMBL9681660

CC#C[Si](C)(C)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP1B1 Q16678 1/20 0.33
NR1H2 P55055 2/20 0.31
NR1H3 Q13133 2/20 0.31
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.30
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3947297 0.87 ESR1 (0.42) ESR1ESR2CYP1A2NR1H2NR1H3
SCHEMBL12191034 0.80 ESR1 (0.38) ESR1ESR2CYP1A1CYP1A2CYP1B1
SCHEMBL12477035 0.80 ESR1 (0.38) ESR1ESR2CYP1A2NR1H2NR1H3
SCHEMBL8135936 0.78 ESR1 (0.37) ESR1ESR2NR1H2NR1H3
SCHEMBL22449371 0.78 ESR1 (0.37) ESR1ESR2NR1H2NR1H3MAPT
SCHEMBL17536636 0.76 APP (0.48) ESR1ESR2CYP1A1CYP1A2CYP1B1
SCHEMBL17552578 0.75 NPC1 (0.35) CYP1A2
SCHEMBL3956326 0.75 ESR1 (0.34) ESR1ESR2NR1H2NR1H3
SCHEMBL17552569 0.75 ESR1 (0.34) ESR1ESR2CYP1A2MAPT
SCHEMBL27795201 0.74 ALDH1A1 (0.39) CYP1A2MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016036685-A1 BASE-CATALYZED SILYLATION OF TERMINIAL ALKYNE C-H BONDS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2016-03-10 WO disclosed
US-20140157452-A1 Plants with Useful Traits and Related Methods BOARD OF REGENTS OF THE UNIVERSITY OF NEBRASKA (US) 2014-06-05 US disclosed
US-5162562-A Preparation of metallated and substituted alkynes AIR PRODUCTS AND CHEMICALS, INC. (US) 1992-11-10 US disclosed
US-5062998-A Preparation of metallated and substituted alkynes AIR PRODUCTS AND CHEMICALS, INC. (US) 1991-11-05 US disclosed
EP-0245516-A1 POLYMER MEMBRANE FOR SEPARATING LIQUID MIXTURE SAGAMI CHEMICAL RESEARCH CENTER (JP) 1987-11-19 EP disclosed