SCHEMBL9681773

SCHEMBL9681773

CCc1ccc(OC)c(CNc2cc(CC)c(CO)[nH]c2=O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.38
KDM4E B2RXH2 5/20 0.38
RECQL P46063 2/20 0.38
APAF1 O14727 1/20 0.38
HTT P42858 3/20 0.38
NPSR1 Q6W5P4 2/20 0.38
GAA P10253 3/20 0.37
LMNA P02545 2/20 0.37
MAPK1 P28482 2/20 0.37
GFER P55789 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TSHR P16473 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
ALDH1A1 P00352 3/20 0.34
HPGD P15428 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846318 0.89 MAPT (0.38) MAPTKDM4ERECQLAPAF1HTT
SCHEMBL9164330 0.85 MAPT (0.41) MAPTKDM4ERECQLAPAF1HTT
SCHEMBL9680853 0.84 MAPT (0.38) MAPTKDM4ERECQLAPAF1HTT
SCHEMBL9680861 0.80 SLC2A1 (0.38) MAPTKDM4ERECQLAPAF1GAA
SCHEMBL9681442 0.79 KDM4E (0.36) MAPTKDM4ERECQLAPAF1IDH1
SCHEMBL9682808 0.79 PDE10A (0.34) MAPTKDM4ERECQLAPAF1LMNA
SCHEMBL9682064 0.75 MAPT (0.34) MAPTKDM4ERECQLAPAF1GAA
SCHEMBL9680359 0.75 MAPT (0.34) MAPTKDM4ERECQLAPAF1GAA
SCHEMBL9681915 0.75 PDE10A (0.40) MAPTKDM4ERECQLAPAF1HTT
SCHEMBL9681299 0.74 MAPT (0.35) MAPTKDM4ERECQLAPAF1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP claimed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed