SCHEMBL9682808

SCHEMBL9682808

CCc1cnc(CNc2cc(CC)c(CO)[nH]c2=O)c(OC)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 8/20 0.34
PDE4D Q08499 1/20 0.33
KDM4E B2RXH2 3/20 0.32
MAPT P10636 2/20 0.32
APAF1 O14727 1/20 0.32
RECQL P46063 1/20 0.32
ABL1 P00519 1/20 0.31
SRC P12931 1/20 0.31
DPP4 P27487 1/20 0.31
POLB P06746 3/20 0.31
ASPH Q12797 1/20 0.31
KDM8 Q8N371 1/20 0.31
GMNN O75496 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
GABRA1 P14867 1/20 0.31
TSHR P16473 1/20 0.31
GABRG2 P18507 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681425 0.84 CYP2C9 (0.33) PDE10AKDM4EMAPTAPAF1RECQL
SCHEMBL9682064 0.81 MAPT (0.34) PDE10AKDM4EMAPTAPAF1RECQL
SCHEMBL9680359 0.81 MAPT (0.34) PDE10AKDM4EMAPTAPAF1RECQL
SCHEMBL9681773 0.79 MAPT (0.38) KDM4EMAPTAPAF1RECQLALDH1A1
SCHEMBL9681442 0.79 KDM4E (0.36) PDE10AKDM4EMAPTAPAF1RECQL
SCHEMBL9681915 0.78 PDE10A (0.40) PDE10AKDM4EMAPTAPAF1RECQL
SCHEMBL9681383 0.78 NPC1 (0.34) KDM4EMAPTAPAF1RECQLPOLB
SCHEMBL9682084 0.78 MAPT (0.36) KDM4EMAPTAPAF1RECQLPOLB
SCHEMBL9680853 0.77 MAPT (0.38) KDM4EMAPTAPAF1RECQLALDH1A1
SCHEMBL9680861 0.73 SLC2A1 (0.38) KDM4EMAPTAPAF1RECQLPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP claimed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed